Synthesis and bradykinin inhibitory activity of novel non-peptide compounds, and evaluation of in vivo analgesic activity (English)
- New search for: Kam, Yoo Lim
- New search for: Rhee, Hee-Kyung
- New search for: Kim, Hwa-Jung
- New search for: Back, Seung Keun
- New search for: Na, Heung Sik
- New search for: Choo, Hea-Young Park
- New search for: Kam, Yoo Lim
- New search for: Rhee, Hee-Kyung
- New search for: Kim, Hwa-Jung
- New search for: Back, Seung Keun
- New search for: Na, Heung Sik
- New search for: Choo, Hea-Young Park
In:
Bioorganic and Medicinal Chemistry
;
18
, 6
;
2327-2336
;
2010
-
ISSN:
- Article (Journal) / Electronic Resource
-
Title:Synthesis and bradykinin inhibitory activity of novel non-peptide compounds, and evaluation of in vivo analgesic activity
-
Contributors:Kam, Yoo Lim ( author ) / Rhee, Hee-Kyung ( author ) / Kim, Hwa-Jung ( author ) / Back, Seung Keun ( author ) / Na, Heung Sik ( author ) / Choo, Hea-Young Park ( author )
-
Published in:Bioorganic and Medicinal Chemistry ; 18, 6 ; 2327-2336
-
Publisher:
-
Publication date:2010-01-20
-
Size:10 pages
-
ISSN:
-
DOI:
-
Type of media:Article (Journal)
-
Type of material:Electronic Resource
-
Language:English
-
Keywords:
-
Source:
Table of contents – Volume 18, Issue 6
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 2067
-
Graphical contents list| 2010
- 2076
-
Structural basis for the design of novel Schiff base metal chelate inhibitors of trypsinIyaguchi, Daisuke / Kawano, Susumu / Takada, Kazuki / Toyota, Eiko et al. | 2010
- 2081
-
Synthesis of theophylline derivatives and study of their activity as antagonists at adenosine receptorsHierrezuelo, Jesús / Manuel López-Romero, J. / Rico, Rodrigo / Brea, José / Isabel Loza, M. / Cai, Chengzhi / Algarra, Manuel et al. | 2010
- 2089
-
Synthesis and biological evaluation of 2′,5′-dimethoxychalcone derivatives as microtubule-targeted anticancer agentsTu, Huang-Yao / Huang, A-Mei / Hour, Tzyh-Chyuan / Yang, Shyh-Chyun / Pu, Yeong-Shiau / Lin, Chun-Nan et al. | 2010
- 2089
-
Synthesis and biological evaluation of 2prime,5prime-dimethoxychalcone derivatives as microtubule-targeted anticancer agentsTu, H. Y. / Huang, A. M. / Hour, T. C. / Yang, S. C. / Pu, Y. S. / Lin, C. N. et al. | 2010
- 2099
-
Synthesis and in vitro biological evaluation of carbon-11-labeled quinoline derivatives as new candidate PET radioligands for cannabinoid CB2 receptor imagingGao, Mingzhang / Wang, Min / Miller, Kathy D. / Hutchins, Gary D. / Zheng, Qi-Huang et al. | 2010
- 2107
-
Design and synthesis of novel series of pyrrole based chemotypes and their evaluation as selective aldose reductase inhibitors. A case of bioisosterism between a carboxylic acid moiety and that of a tetrazolePegklidou, Kyriaki / Koukoulitsa, Catherine / Nicolaou, Ioannis / Demopoulos, Vassilis J. et al. | 2010
- 2115
-
Chemical biology studies on norrisolideGuizzunti, Gianni / Brady, Thomas P. / Fischer, Derek / Malhotra, Vivek / Theodorakis, Emmanuel A. et al. | 2010
- 2123
-
Efflux-mediated bis-indole resistance in Staphylococcus aureus reveals differential substrate specificities for MepA and MepROpperman, Timothy J. / Williams, John D. / Houseweart, Chad / Panchal, Rekha G. / Bavari, Sina / Peet, Norton P. / Moir, Donald T. / Bowlin, Terry L. et al. | 2010
- 2131
-
Gentisides A and B, two new neuritogenic compounds from the traditional Chinese medicine Gentiana rigescens FranchGao, Lijuan / Li, Jinyou / Qi, Jianhua et al. | 2010
- 2135
-
SAR and molecular mechanism study of novel acylhydrazone compounds targeting HIV-1 CAJin, Yinxue / Tan, Zhiwu / He, Meizi / Tian, Baohe / Tang, Shixing / Hewlett, Indira / Yang, Ming et al. | 2010
- 2141
-
Exploration of inhibitors for diaminopimelate aminotransferaseFan, Chenguang / Clay, Matthew D. / Deyholos, Michael K. / Vederas, John C. et al. | 2010
- 2152
-
Alstiphyllanines E–H, picraline and ajmaline-type alkaloids from Alstonia macrophylla inhibiting sodium glucose cotransporterArai, Hiroko / Hirasawa, Yusuke / Rahman, Abdul / Kusumawati, Idha / Zaini, Noor Cholies / Sato, Seizo / Aoyama, Chihiro / Takeo, Jiro / Morita, Hiroshi et al. | 2010
- 2159
-
Carbonic anhydrase inhibitors. Inhibition of mammalian isoforms I–XIV with a series of natural product polyphenols and phenolic acidsInnocenti, Alessio / Beyza Öztürk Sarıkaya, S. / Gülçin, İlhami / Supuran, Claudiu T. et al. | 2010
- 2165
-
A class of novel Schiff’s bases: Synthesis, therapeutic action for chronic pain, anti-inflammation and 3D QSAR analysisZhou, Yinjian / Zhao, Ming / Wu, Yingting / Li, Chunyu / Wu, Jianhui / Zheng, Meiqing / Peng, Li / Peng, Shiqi et al. | 2010
- 2173
-
Acetylcholinesterase inhibitors from the toadstool Cortinarius infractusGeissler, Torsten / Brandt, Wolfgang / Porzel, Andrea / Schlenzig, Dagmar / Kehlen, Astrid / Wessjohann, Ludger / Arnold, Norbert et al. | 2010
- 2178
-
Novel C-aryl glucoside SGLT2 inhibitors as potential antidiabetic agents: 1,3,4-Thiadiazolylmethylphenyl glucoside congenersLee, Junwon / Lee, Sung-Han / Seo, Hee Jeong / Son, Eun-Jung / Lee, Suk Ho / Jung, Myung Eun / Lee, MinWoo / Han, Ho-Kyun / Kim, Jeongmin / Kang, Jahyo et al. | 2010
- 2195
-
2-Amino-5-benzoyl-4-phenylthiazoles: Development of potent and selective adenosine A1 receptor antagonistsScheiff, Anja B. / Yerande, Swapnil G. / El-Tayeb, Ali / Li, Wenjin / Inamdar, Gajanan S. / Vasu, Kamala K. / Sudarsanam, Vasudevan / Müller, Christa E. et al. | 2010
- 2204
-
In silico search for multi-target anti-inflammatories in Chinese herbs and formulasEhrman, Thomas M. / Barlow, David J. / Hylands, Peter J. et al. | 2010
- 2219
-
Cytotoxic 2-benzylidene-6-(nitrobenzylidene)cyclohexanones which display substantially greater toxicity for neoplasms than non-malignant cellsDas, Umashankar / Doroudi, Alireza / Inci Gul, H. / Pati, Hari N. / Kawase, Masami / Sakagami, Hiroshi / Chu, Qing / Stables, James P. / Dimmock, Jonathan R. et al. | 2010
- 2225
-
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite speciesPrado-Prado, Francisco J. / García-Mera, Xerardo / González-Díaz, Humberto et al. | 2010
- 2232
-
Differential binding of phenothiazine urea derivatives to wild-type human cholinesterases and butyrylcholinesterase mutantsDarvesh, Sultan / Pottie, Ian R. / Darvesh, Katherine V. / McDonald, Robert S. / Walsh, Ryan / Conrad, Sarah / Penwell, Andrea / Mataija, Diane / Martin, Earl et al. | 2010
- 2245
-
Synthesis of 2-(thienyl-2-yl or -3-yl)-4-furyl-6-aryl pyridine derivatives and evaluation of their topoisomerase I and II inhibitory activity, cytotoxicity, and structure–activity relationshipThapa, Pritam / Karki, Radha / Choi, Hoyoung / Choi, Jae Hun / Yun, Minho / Jeong, Byeong-Seon / Jung, Mi-Ja / Nam, Jung Min / Na, Younghwa / Cho, Won-Jea et al. | 2010
- 2255
-
Synthesis, radiofluorination, and hypoxia-selective studies of FRAZ: A configurational and positional analogue of the clinical hypoxia marker, [18F]-FAZAKumar, Piyush / Naimi, Ebrahim / McEwan, Alexander J. / Wiebe, Leonard I. et al. | 2010
- 2265
-
Synthesis and kinetic analysis of some phosphonate analogs of cyclophostin as inhibitors of human acetylcholinesteraseDutta, Supratik / Malla, Raj K. / Bandyopadhyay, Saibal / Spilling, Christopher D. / Dupureur, Cynthia M. et al. | 2010
- 2275
-
Structural-based design and synthesis of novel 9-deazaguanine derivatives having a phosphate mimic as multi-substrate analogue inhibitors for mammalian PNPsHikishima, Sadao / Hashimoto, Mariko / Magnowska, Lucyna / Bzowska, Agnieszka / Yokomatsu, Tsutomu et al. | 2010
- 2285
-
Potent DNA-directed alkylating agents: Synthesis and biological activity of phenyl N-mustard–quinoline conjugates having a urea or hydrazinecarboxamide linkerKakadiya, Rajesh / Dong, Huajin / Kumar, Amit / Narsinh, Dodia / Zhang, Xiuguo / Chou, Ting-Chao / Lee, Te-Chang / Shah, Anamik / Su, Tsann-Long et al. | 2010
- 2300
-
Carbonic anhydrase activators. The first activation study of a coral secretory isoform with amino acids and aminesBertucci, Anthony / Zoccola, Didier / Tambutté, Sylvie / Vullo, Daniela / Supuran, Claudiu T. et al. | 2010
- 2304
-
Pharmacophore modeling, resistant mutant isolation, docking, and MM-PBSA analysis: Combined experimental/computer-assisted approaches to identify new inhibitors of the bovine viral diarrhea virus (BVDV)Tonelli, Michele / Boido, Vito / Colla, Paolo La / Loddo, Roberta / Posocco, Paola / Paneni, Maria Silvia / Fermeglia, Maurizio / Pricl, Sabrina et al. | 2010
- 2317
-
Design, synthesis and evaluation of (E)-a-benzylthio chalcones as novel inhibitors of BCR-ABL kinaseReddy, M. V. / Pallela, V. R. / Cosenza, S. C. / Mallireddigari, M. R. / Patti, R. / Bonagura, M. / Truongcao, M. / Akula, B. / Jatiani, S. S. / Reddy, E. P. et al. | 2010
- 2317
-
Design, synthesis and evaluation of (E)-α-benzylthio chalcones as novel inhibitors of BCR-ABL kinaseReddy, M.V. Ramana / Pallela, Venkat R. / Cosenza, Stephen C. / Mallireddigari, Muralidhar R. / Patti, Revathi / Bonagura, Marie / Truongcao, May / Akula, Balaiah / Jatiani, Shashidhar S. / Reddy, E. Premkumar et al. | 2010
- 2327
-
Synthesis and bradykinin inhibitory activity of novel non-peptide compounds, and evaluation of in vivo analgesic activityKam, Yoo Lim / Rhee, Hee-Kyung / Kim, Hwa-Jung / Back, Seung Keun / Na, Heung Sik / Choo, Hea-Young Park et al. | 2010
- 2337
-
Melanogenesis inhibitors from the desert plant Anastatica hierochuntica in B16 melanoma cellsNakashima, Souichi / Matsuda, Hisashi / Oda, Yoshimi / Nakamura, Seikou / Xu, Fengming / Yoshikawa, Masayuki et al. | 2010
- 2346
-
Corrigendum to “Inhibitors of human tyrosyl-DNA phospodiesterase (hTdp1) developed by virtual screening using ligand-based pharmacophores” [Bioorg. Med. Chem. 18 (2010) 182–189]Weidlich, Iwona E. / Dexheimer, Thomas / Marchand, Christophe / Antony, Smitha / Pommier, Yves / Nicklaus, Marc C. et al. | 2010
- 2347
-
Virtual screening using ligand-based pharmacophores for inhibitors of human tyrosyl-DNA phospodiesterase (hTdp1)Weidlich, Iwona E. / Dexheimer, Thomas S. / Marchand, Christophe / Antony, Smitha / Pommier, Yves / Nicklaus, Marc C. et al. | 2010
- IFC
-
Editorial board| 2010