Synthetic bioactive olivetol-related amides: The influence of the phenolic group in cannabinoid receptor activity (English)
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- New search for: Pertwee, Roger G.
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- New search for: Boccella, Serena
- New search for: Cascio, Maria Grazia
- New search for: De Petrocellis, Luciano
- New search for: Frosini, Maria
- New search for: Gado, Francesca
- New search for: Ligresti, Alessia
- New search for: Luongo, Livio
- New search for: Marini, Pietro
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In:
Bioorganic and Medicinal Chemistry
;
28
, 11
;
2020
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ISSN:
- Article (Journal) / Electronic Resource
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Title:Synthetic bioactive olivetol-related amides: The influence of the phenolic group in cannabinoid receptor activity
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Contributors:Brizzi, Antonella ( author ) / Aiello, Francesca ( author ) / Boccella, Serena ( author ) / Cascio, Maria Grazia ( author ) / De Petrocellis, Luciano ( author ) / Frosini, Maria ( author ) / Gado, Francesca ( author ) / Ligresti, Alessia ( author ) / Luongo, Livio ( author ) / Marini, Pietro ( author )
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Published in:Bioorganic and Medicinal Chemistry ; 28, 11
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Publisher:
- New search for: Elsevier Ltd
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Publication date:2020-04-16
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ISSN:
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DOI:
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Type of media:Article (Journal)
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Type of material:Electronic Resource
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Language:English
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Keywords:
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Source:
Table of contents – Volume 28, Issue 11
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
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Synthesis and structure-activity relationships of thieno[2,3-d]pyrimidines as atypical protein kinase C inhibitors to control retinal vascular permeability and cytokine-induced edemaLiu, Xuwen / Wilson, Michael W. / Liu, Kun / Lee, Pil / Yeomans, Larisa / Hagen, Susan E. / Lin, Cheng-Mao / Wen, Bo / Sun, Duxin / White, Andrew D. et al. | 2020
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Cytotoxicity of 4-substituted quinoline derivatives: Anticancer and antileishmanial potentialCosta, Claudia A. / Lopes, Rayssa M. / Ferraz, Leticia S. / Esteves, Gabriela N.N. / Di Iorio, Juliana F. / Souza, Aline A. / de Oliveira, Isadora M. / Manarin, Flavia / Judice, Wagner A.S. / Stefani, Helio A. et al. | 2020
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Editorial Board| 2020
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Graphical abstract TOC| 2020
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Synthesis and evaluation of 7-azaindole derivatives bearing benzocycloalkanone motifs as protein kinase inhibitorsQhobosheane, Malikotsi A. / Legoabe, Lesetja J. / Josselin, Béatrice / Bach, Stéphane / Ruchaud, Sandrine / Petzer, Jacobus P. / Beteck, Richard M. et al. | 2020
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A novel Golgi mannosidase inhibitor: Molecular design, synthesis, enzyme inhibition, and inhibition of spheroid formationKoyama, Ryosuke / Kano, Yui / Kikushima, Kaori / Mizutani, Ayaka / Soeda, Yuta / Miura, Kazuki / Hirano, Takako / Nishio, Toshiyuki / Hakamata, Wataru et al. | 2020
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Design and synthesis of 1,3-benzothiazinone derivatives as potential anti-inflammatory agentsLi, Junfang / Fan, Xiaohong / Deng, Jiedan / Liang, Yan / Ma, Shumeng / Lu, Yingmei / Zhang, Jian / Shi, Tao / Tan, Wen / Wang, Zhen et al. | 2020
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Syntheses and pharmacokinetic evaluations of four metabolites of 2-(4-(2-((1H-benzo[d]imidazol-2-yl)thio)ethyl)piperazin-1-yl)-N-(6-methyl-2,4-bis-(methylthio)pyridin-3-yl)acetamide hydrochloride [K-604], an acyl-CoA:cholesterol O-acyltransferase-1 inhibitorShibuya, Kimiyuki / Miura, Toru / Ohgiya, Tadaaki / Omichi, Kozo / Tsunenari, Yoshihiko et al. | 2020
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Enzymatic synthesis of biphenyl-DNA oligonucleotidesRöthlisberger, Pascal / Levi-Acobas, Fabienne / Leumann, Christian J. / Hollenstein, Marcel et al. | 2020
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Inhibition of bacterial growth and galactosyltransferase activity of WbwC by α, ω-bis(3-alkyl-1H-imidazolium)alkane salts: Effect of varying carbon contentKocev, Alexander / Melamed, Jacob / Wang, Shuo / Kong, Xianqi / Vlahakis, Jason Z. / Xu, Yaozu / Szarek, Walter A. / Brockhausen, Inka et al. | 2020
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Secondary metabolites from Isodon ternifolius (D. Don) Kudo and their anticancer activity as DNA topoisomerase IB and Tyrosyl-DNA phosphodiesterase 1 inhibitorsZhang, Hong-Li / Zhang, Yu / Yan, Xue-Long / Xiao, Long-Gao / Hu, De-Xuan / Yu, Qian / An, Lin-Kun et al. | 2020
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Microbial transformation of glycyrrhetinic acid derivatives by Bacillus subtilis ATCC 6633 and Bacillus megaterium CGMCC 1.1741Shen, Pingping / Zhang, Jian / Zhu, Yuyuan / Wang, Wei / Yu, Boyang / Wang, Weiwei et al. | 2020
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Exploratory studies on CA-15L, an anti-HIV active HIV-1 capsid fragmentTsuji, Kohei / Owusu, Kofi Baffour-Awuah / Kobayakawa, Takuya / Wang, Rongyi / Fujino, Masayuki / Kaneko, Moemi / Yamamoto, Naoki / Murakami, Tsutomu / Tamamura, Hirokazu et al. | 2020
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Discovery of novel, potent, and orally bioavailable pyrido[2,3-d][1]benzazepin-6-one antagonists for parathyroid hormone receptor 1Arai, Yoshikazu / Kiyotsuka, Yohei / Kagechika, Katsuji / Nishi, Tatsuya / Inui, Masaharu / Nagamochi, Masatoshi / Oyama, Kazunori / Izumi, Masanori et al. | 2020
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An aza-nucleoside, fragment-like inhibitor of the DNA repair enzyme alkyladenine glycosylase (AAG)Mas Claret, Eduard / Al Yahyaei, Balqees / Chu, Shuyu / Elliott, Ruan M. / Imperato, Manuel / Lopez, Arnaud / Meira, Lisiane B. / Howlin, Brendan J. / Whelligan, Daniel K. et al. | 2020
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Design and synthesis of novel pyrrolo[2,3-b]pyridine derivatives targeting V600EBRAFAbdel-Maksoud, Mohammed S. / Ali, Eslam M.H. / Ammar, Usama M. / Mersal, Karim I. / Yoo, Kyung Ho / Oh, Chang-Hyun et al. | 2020
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Discovery of a new potent inhibitor of mushroom tyrosinase (Agaricus bisporus) containing 4-(4-hydroxyphenyl)piperazin-1-yl moietyDe Luca, Laura / Germanò, Maria Paola / Fais, Antonella / Pintus, Francesca / Buemi, Maria Rosa / Vittorio, Serena / Mirabile, Salvatore / Rapisarda, Antonio / Gitto, Rosaria et al. | 2020
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Graphical Abstract Contents Continued| 2020
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Optimization and biological evaluation of imidazopyridine derivatives as a novel scaffold for γ-secretase modulators with oral efficacy against cognitive deficits in Alzheimer’s disease model miceSekioka, Ryuichi / Honda, Shugo / Akashiba, Hiroki / Yarimizu, Junko / Mitani, Yasuyuki / Yamasaki, Shingo et al. | 2020
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Progress towards drug discovery for Friedreich’s Ataxia: Identifying synthetic oligonucleotides that more potently activate expression of human frataxin proteinShen, Xiulong / Wong, Johnathan / Prakash, Thahza P. / Rigo, Frank / Li, Yanjie / Napierala, Marek / Corey, David R. et al. | 2020
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Syntheses, in vitro α-amylase and α-glucosidase dual inhibitory activities of 4-amino-1,2,4-triazole derivatives their molecular docking and kinetic studiesYeye, Emmanuel Oloruntoba / Kanwal / Mohammed Khan, Khalid. / Chigurupati, Sridevi / Wadood, Abdul / Ur Rehman, Ashfaq / Perveen, Shahnaz / Kannan Maharajan, Mari / Shamim, Shahbaz / Hameed, Shehryar et al. | 2020
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Structure-activity relationship studies on the inhibition of the bacterial translation of novel Odilorhabdins analoguesLoza, Einars / Sarciaux, Matthieu / Ikaunieks, Martins / Katkevics, Martins / Kukosha, Tatyana / Trufilkina, Nadezhda / Ryabova, Victoria / Shubin, Kirill / Pantel, Lucile / Serri, Marine et al. | 2020
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Synthesis and cytotoxic effects of 2-thio-3,4-dihydroquinazoline derivatives as novel T-type calcium channel blockersNam, Yunchan / Ryu, Ki Deok / Jang, Changyoung / Moon, Yoon Hyoung / Kim, Misong / Ko, Dohyeong / Chung, Kyung-Sook / Gandini, Maria A. / Lee, Kyung-Tae / Zamponi, Gerald W. et al. | 2020
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Synthetic bioactive olivetol-related amides: The influence of the phenolic group in cannabinoid receptor activityBrizzi, Antonella / Aiello, Francesca / Boccella, Serena / Cascio, Maria Grazia / De Petrocellis, Luciano / Frosini, Maria / Gado, Francesca / Ligresti, Alessia / Luongo, Livio / Marini, Pietro et al. | 2020
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Induction of enantio-selective apoptosis in human leukemia HL-60 cells by (S)-erypoegin K, an isoflavone isolated from Erythrina poeppigianaHikita, Kiyomi / Saigusa, Satomi / Takeuchi, Yuto / Matsuyama, Haruka / Nagai, Rina / Kato, Kuniki / Murata, Tomiyasu / Tanaka, Hitoshi / Wagh, Yogesh S. / Asao, Naoki et al. | 2020
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Design, synthesis and acaricidal activities of Cyflumetofen analogues based on carbon-silicon isosteric replacementZhou, Cong / Cheng, Jiagao / Beadle, Ryan / Earley, Fergus G. / Li, Zhong / Maienfisch, Peter et al. | 2020
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Synthesis, state-of-the-art NMR-binding and molecular modeling study of new benzimidazole core derivatives as Pin1 inhibitors: Targeting breast cancerNashaat, Samira / Henen, Morkos A. / El-Messery, Shahenda M. / Eisa, Hassan et al. | 2020
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Deuteration of the farnesyl terminal methyl groups of δ-tocotrienol and its effects on the metabolic stability and ability of inducing G-CSF productionLiu, Xingui / Gao, Zhengya / Fu, Qiang / Song, Lin / Zhang, Peiyi / Zhang, Xuan / Hendrickson, Howard / Crooks, Peter A. / Zhou, Daohong / Zheng, Guangrong et al. | 2020
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Structural modifications of indolinones bearing a pyrrole moiety and discovery of a multi-kinase inhibitor with potent antitumor activityQin, Mingze / Tian, Ye / Han, Xiao / Cao, Qi / Zheng, Shuaishuai / Liu, Chunyang / Wu, Xia / Liu, Lei / Meng, Yangyang / Wang, Xiaobo et al. | 2020
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Benzoxepinones: A new isoform-selective class of tumor associated carbonic anhydrase inhibitorsGrandane, Aiga / Nocentini, Alessio / Werner, Thomas / Zalubovskis, Raivis / Supuran, Claudiu T. et al. | 2020