Synthesis and biological evaluation of a technetium-99m(I)-tricarbonyl-labelled phenyltropane derivative (English)
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In:
Bioorganic & medicinal chemistry letters
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16
, 2
; 382-386
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2006
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ISSN:
- Article (Journal) / Print
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Title:Synthesis and biological evaluation of a technetium-99m(I)-tricarbonyl-labelled phenyltropane derivative
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Contributors:
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Published in:Bioorganic & medicinal chemistry letters ; 16, 2 ; 382-386
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Publisher:
- New search for: Elsevier
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Place of publication:Amsterdam [u.a.]
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Publication date:2006
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Type of media:Article (Journal)
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Type of material:Print
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Language:English
- New search for: 35.70 / 44.33 / 44.42
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Source:
Table of contents – Volume 16, Issue 2
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 235
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Graphical contents list| 2005
- 248
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Non-covalent modification of the heme-pocket of apomyoglobin by a 1,10-phenanthroline derivativeHitomi, Yutaka / Mukai, Hidefumi / Yoshimura, Hideaki / Tanaka, Tsunehiro / Funabiki, Takuzo et al. | 2005
- 252
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Synthesis and biological evaluation of novel pyrrolo[2,1-c][1,4]benzodiazepine prodrugs for use in antibody-directed enzyme prodrug therapyMasterson, Luke A. / Spanswick, Victoria J. / Hartley, John A. / Begent, Richard H. / Howard, Philip W. / Thurston, David E. et al. | 2005
- 257
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Design, synthesis, and vasorelaxant and platelet antiaggregatory activities of coumarin#8211resveratrol hybridsVilar, Santiago et al. | 2006
- 257
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Design, synthesis, and vasorelaxant and platelet antiaggregatory activities of coumarin–resveratrol hybridsVilar, Santiago / Quezada, Elías / Santana, Lourdes / Uriarte, Eugenio / Yánez, Matilde / Fraiz, Nuria / Alcaide, Carlos / Cano, Ernesto / Orallo, Francisco et al. | 2005
- 262
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Pyrazoloheteroaryls: Novel p38α MAP kinase inhibiting scaffolds with oral activityRevesz, Laszlo / Blum, Ernst / Di Padova, Franco E. / Buhl, Thomas / Feifel, Roland / Gram, Hermann / Hiestand, Peter / Manning, Ute / Neumann, Ulf / Rucklin, Gerard et al. | 2005
- 262
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Pyrazoloheteroaryls: Novel p38#945 MAP kinase inhibiting scaffolds with oral activityRevesz, Laszlo et al. | 2006
- 267
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Biphenyl-4-ylcarbamoyl thiophene carboxylic acids as potent DHODH inhibitorsLeban, Johann / Kralik, Martin / Mies, Jan / Baumgartner, Roland / Gassen, Michael / Tasler, Stefan et al. | 2005
- 271
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Benzylprotected aromatic phosphonic acids for anchoring peptides on titaniumAuernheimer, Jörg / Kessler, Horst et al. | 2005
- 274
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Specific volume and compressibility of human serum albumin–polyanion complexesHianik, Tibor / Poniková, Slavomíra / Bágel’ová, Jaroslava / Antalík, Marián et al. | 2005
- 274
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Specific volume and compressibility of human serum albumin#8211polyanion complexesHianik, Tibor et al. | 2006
- 280
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4-Substituted cyclohexyl sulfones as potent, orally active γ-secretase inhibitorsChurcher, Ian / Beher, Dirk / Best, Jonathan D. / Castro, José L. / Clarke, Earl E. / Gentry, Amy / Harrison, Timothy / Hitzel, Laure / Kay, Euan / Kerrad, Sonia et al. | 2005
- 280
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4-Substituted cyclohexyl sulfones as potent, orally active #947-secretase inhibitorsChurcher, Ian et al. | 2006
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- 288
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5-Heteroatom substituted pyrazoles as canine COX-2 inhibitors. Part 1: Structure#8211activity relationship studies of 5-alkylamino pyrazoles and discovery of a potent, selective, and orally active analogSakya, Subas M. et al. | 2006
- 293
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4-Hydroxyisoleucine an unusual amino acid as antidyslipidemic and antihyperglycemic agentNarender, Tadigoppula / Puri, Anju / Shweta / Khaliq, Tanvir / Saxena, Rashmi / Bhatia, Geetika / Chandra, Ramesh et al. | 2005
- 297
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Substituted indanylacetic acids as PPAR-α–γ activatorsLowe, Derek B. / Bifulco, Neil / Bullock, William H. / Claus, Thomas / Coish, Philip / Dai, Miao / Dela Cruz, Fernando E. / Dickson, David / Fan, Dongping / Hoover-Litty, Helana et al. | 2005
- 297
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Substituted indanylacetic acids as PPAR-#945#8211#947 activatorsLowe, Derek B. et al. | 2006
- 302
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Novel 1,3-dipropyl-8-(1-heteroarylmethyl-1H-pyrazol-4-yl)-xanthine derivatives as high affinity and selective A2B adenosine receptor antagonistsElzein, Elfatih / Kalla, Rao / Li, Xiaofen / Perry, Thao / Parkhill, Eric / Palle, Venkata / Varkhedkar, Vaibahv / Gimbel, Art / Zeng, Dewan / Lustig, David et al. | 2005
- 307
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A new chemical tool for exploring the physiological function of the PDE2 isozymeChambers, Robert J. / Abrams, Kristin / Garceau, Norman Y. / Kamath, Ajith V. / Manley, Christopher M. / Lilley, Susan C. / Otte, Douglas A. / Scott, Dennis O. / Sheils, Alissa L. / Tess, David A. et al. | 2005
- 311
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Synthesis and biological evaluation of biphenylsulfonamide carboxylate aggrecanase-1 inhibitorsXiang, Jason S. / Hu, Yonghan / Rush, Thomas S. / Thomason, Jennifer R. / Ipek, Manus / Sum, Phaik-Eng / Abrous, Leila / Sabatini, Joshua J. / Georgiadis, Katy / Reifenberg, Erica et al. | 2005
- 317
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Synthesis and biological activities of nucleoside–estradiol conjugatesAli, Hasrat / Ahmed, Naseem / Tessier, Guillaume / van Lier, Johan E. et al. | 2005
- 317
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Synthesis and biological activities of nucleoside#8211estradiol conjugatesAli, Hasrat et al. | 2006
- 320
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Leptostatin: A synthetic hybrid of the cytotoxic polyketides callystatin A and leptomycin BMarshall, James A. / Mikowski, Ann M. / Bourbeau, Matthew P. / Schaaf, Gregory M. / Valeriote, Frederick et al. | 2005
- 324
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New tyrosinase inhibitors selected by atomic linear indices-based classification modelsCasañola-Martín, Gerardo M. / Khan, Mahmud Tareq Hassan / Marrero-Ponce, Yovani / Ather, Arjumand / Sultankhodzhaev, Mukhlis N. / Torrens, Francisco et al. | 2005
- 331
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PET imaging and optical imaging with d-luciferin [11C]methyl ester and d-luciferin [11C]methyl ether of luciferase gene expression in tumor xenografts of living miceWang, Ji-Quan / Pollok, Karen E. / Cai, Shanbao / Stantz, Keith M. / Hutchins, Gary D. / Zheng, Qi-Huang et al. | 2005
- 338
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Structure-based design of novel groups for use in the P1 position of thrombin inhibitor scaffolds. Part 1: Weakly basic azolesIsaacs, Richard C.A. / Solinsky, Mark G. / Cutrona, Kellie J. / Newton, Christina L. / Naylor-Olsen, Adel M. / Krueger, Julie A. / Lewis, S. Dale / Lucas, Bobby J. et al. | 2005
- 343
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Design, synthesis and structure–activity relationships of new phosphinate inhibitors of MurDŠtrancar, Katja / Blanot, Didier / Gobec, Stanislav et al. | 2005
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Design, synthesis and structure#8211activity relationships of new phosphinate inhibitors of MurD| 2006
- 349
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Discovery of N-(2-aryl-cyclohexyl) substituted spiropiperidines as a novel class of GlyT1 inhibitorsPinard, Emmanuel / Ceccarelli, Simona M. / Stalder, Henri / Alberati, Daniela et al. | 2005
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Discovery of N-(2-hydroxy-2-aryl-cyclohexyl) substituted spiropiperidines as GlyT1 antagonists with improved pharmacological profileCeccarelli, Simona M. / Pinard, Emmanuel / Stalder, Henri / Alberati, Daniela et al. | 2005
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Dipeptide-based highly potent doxorubicin antibody conjugatesJeffrey, Scott C. / Nguyen, Minh T. / Andreyka, Jamie B. / Meyer, Damon L. / Doronina, Svetlana O. / Senter, Peter D. et al. | 2005
- 363
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Biomimetic synthesis and ultrastructural characterization of a zerovalent gold#8211hydroxyapatite compositeGupta, Yogita et al. | 2006
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Biomimetic synthesis and ultrastructural characterization of a zerovalent gold–hydroxyapatite compositeGupta, Yogita / Mathur, G.N. / Verma, Sandeep et al. | 2005
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Synthesis and biological activity of the first cyclic biphalin analoguesMollica, Adriano / Davis, Peg / Ma, Shou-Wu / Porreca, Frank / Lai, Josephine / Hruby, Victor J. et al. | 2005
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Potent anti-muscarinic activity in a novel series of quinuclidine derivativesStarck, Jean-Philippe / Talaga, Patrice / Quéré, Luc / Collart, Philippe / Christophe, Bernard / Brutto, Patrick Lo / Jadot, Sophie / Chimmanamada, Dinesh / Zanda, Matteo / Wagner, Alain et al. | 2005
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The identification of potent and selective imidazole-based inhibitors of B-Raf kinaseTakle, Andrew K. / Brown, Murray J.B. / Davies, Susannah / Dean, David K. / Francis, Gerraint / Gaiba, Alessandra / Hird, Alex W. / King, Frank D. / Lovell, Peter J. / Naylor, Antoinette et al. | 2005
- 382
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Synthesis and biological evaluation of a technetium-99m(I)-tricarbonyl-labelled phenyltropane derivativeKieffer, Davy M. / Cleynhens, Bernard J. / Vanbilloen, Hubert P. / Rattat, Dirk / Terwinghe, Christelle Y. / Mortelmans, Luc / Bormans, Guy M. / Verbruggen, Alfons M. et al. | 2005
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Macrolactonization to 10-deoxymethynolide catalyzed by the recombinant thioesterase of the picromycin/methymycin polyketide synthaseHe, Weiguo / Wu, Jiaquan / Khosla, Chaitan / Cane, David E. et al. | 2005
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Instructions to contributors| 2005