1,5-Biaryl pyrrole derivatives as EP1 receptor antagonists. Structure–activity relationships of 6-substituted and 5,6-disubstituted benzoic acid derivatives (English)
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In:
Bioorganic & medicinal chemistry letters
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17
, 4
; 916-920
;
2007
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ISSN:
- Article (Journal) / Print
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Title:1,5-Biaryl pyrrole derivatives as EP1 receptor antagonists. Structure–activity relationships of 6-substituted and 5,6-disubstituted benzoic acid derivatives
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Contributors:
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Published in:Bioorganic & medicinal chemistry letters ; 17, 4 ; 916-920
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Publisher:
- New search for: Elsevier
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Place of publication:Amsterdam [u.a.]
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Publication date:2007
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ISSN:
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ZDBID:
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Type of media:Article (Journal)
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Type of material:Print
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Language:English
- New search for: 35.70 / 44.33 / 44.42
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Source:
Table of contents – Volume 17, Issue 4
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
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Graphical contents list| 2007
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Pharmacophoric features of Pseudomonas aeruginosa deacetylase LpxC inhibitors: An electronic and structural analysisKadam, Rameshwar U. / Chavan, Archana / Roy, Nilanjan et al. | 2006
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Synthesis and biological evaluation of thiazolidine-2-one 1,1-dioxide as inhibitors of Escherichia coli β-ketoacyl-ACP-synthase III (FabH)Alhamadsheh, Mamoun M. / Waters, Norman C. / Huddler, Donald P. / Kreishman-Deitrick, Mara / Florova, Galina / Reynolds, Kevin A. et al. | 2006
- 879
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Synthesis and biological evaluation of thiazolidine-2-one 1,1-dioxide as inhibitors of Escherichia coli b-ketoacyl-ACP-synthase III (FabH)Alhamadsheh, M. M. / Waters, N. C. / Huddler, D. P. / Kreishman-Deitrick, M. / Florova, G. / Reynolds, K. A. et al. | 2007
- 884
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Constrained 7-fluorocarboxychromone-4-aminopiperidine based Melanin-concentrating hormone receptor 1 antagonists: The effects of chirality on substituted indan-1-ylaminesSouers, Andrew J. / Iyengar, Rajesh R. / Judd, Andrew S. / Beno, David W.A. / Gao, Ju / Zhao, Gang / Brune, Michael E. / Napier, James J. / Mulhern, Mathew M. / Lynch, John K. et al. | 2006
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ERβ ligands. Part 5: Synthesis and structure–activity relationships of a series of 4′-hydroxyphenyl-aryl-carbaldehyde oxime derivativesMewshaw, Richard E. / Bowen, S. Marc / Harris, Heather A. / Xu, Zhang B. / Manas, Eric S. / Cohn, Stephen T. et al. | 2006
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ERb ligands. Part 5: Synthesis and structure-activity relationships of a series of 4prime-hydroxyphenyl-aryl-carbaldehyde oxime derivativesMewshaw, R. E. / Bowen, S. M. / Harris, H. A. / Xu, Z. B. / Manas, E. S. / Cohn, S. T. et al. | 2007
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- 916
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1,5-Biaryl pyrrole derivatives as EP1 receptor antagonists. Structure–activity relationships of 6-substituted and 5,6-disubstituted benzoic acid derivativesHall, Adrian / Brown, Susan H. / Chessell, Iain P. / Chowdhury, Anita / Clayton, Nicholas M. / Coleman, Tanya / Giblin, Gerard M.P. / Hammond, Beverley / Healy, Mark P. / Johnson, Matthew R. et al. | 2006
- 921
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Kinetic resolution of (±)-1-phenylethanol in [Bmim][PF6] using high activity preparations of lipasesShah, Shweta / Gupta, Munishwar N. et al. | 2006
- 925
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1,5-Benzodioxepin derivatives as a novel class of muscarinic M3 receptor antagonistsSonda, Shuji / Katayama, Kenichi / Fujio, Masakazu / Sakashita, Hiroshi / Inaba, Kenichi / Asano, Kiyoshi / Akira, Toshiaki et al. | 2006
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The crystal structure, self-assembly, DNA-binding and cleavage studies of the [2]pseudorotaxane composed of cucurbit[6]urilHuo, Fang-Jun / Yin, Cai-Xia / Yang, Pin et al. | 2006
- 937
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Design and synthesis of oxime ethers of α-acyl-β-phenylpropanoic acids as PPAR dual agonistsOon Han, Hee / Hae Kim, Seung / Kim, Kyoung-Hee / Hur, Gwong-Cheung / Joo Yim, Hyeon / Chung, Hee-Kyung / Ho Woo, Sung / Dong Koo, Ki / Lee, Chang-Seok / Sung Koh, Jong et al. | 2006
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Design and synthesis of oxime ethers of a-acyl-b-phenylpropanoic acids as PPAR dual agonistsOon Han, H. / Hae Kim, S. / Kim, K. H. / Hur, G. C. / Joo Yim, H. / Chung, H. K. / Ho Woo, S. / Dong Koo, K. / Lee, C. S. / Sung Koh, J. et al. | 2007
- 942
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Synthesis and antibacterial activities of new quinolone derivatives utilizing 1-azabicyclo[1.1.0]butaneIkee, Yoshifumi / Hashimoto, Kana / Nakashima, Masaaki / Hayashi, Kazuhiko / Sano, Shigeki / Shiro, Motoo / Nagao, Yoshimitsu et al. | 2006
- 946
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Novel fluorescent analogues for transmembrane movement study of polyprenyl phosphatesKoseki, Koichi / Yamashita, Satoshi / Takahashi, Seiji / Koyama, Tanetoshi et al. | 2006
- 951
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5-Propynylamino α-deoxyuridine promotes DNA duplex stabilization of anionic and neutral but not cationic α-oligonucleotidesDeglane, Gaëlle / Morvan, François / Debart, Françoise / Vasseur, Jean-Jacques et al. | 2006
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5-Propynylamino a-deoxyuridine promotes DNA duplex stabilization of anionic and neutral but not cationic a-oligonucleotidesDeglane, G. / Morvan, F. / Debart, F. / Vasseur, J. J. et al. | 2007
- 955
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2-(2,2,2-Trifluoroethyl)-5,6-dichlorobenzimidazole derivatives as potent androgen receptor antagonistsNg, Raymond A. / Guan, Jihua / Alford, Vernon C. Jr. / Lanter, James C. / Allan, George F. / Sbriscia, Tifanie / Lundeen, Scott G. / Sui, Zhihua et al. | 2006
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Synthesis and antimalarial evaluation of a series of piperazinyl flavonesAuffret, Gwenola / Labaied, Mehdi / Frappier, François / Rasoanaivo, Philippe / Grellier, Philippe / Lewin, Guy et al. | 2006
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Inhibitors of the FEZ-1 metallo-b-lactamaseLienard, B. M. / Horsfall, L. E. / Galleni, M. / Frere, J. M. / Schofield, C. J. et al. | 2007
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Inhibitors of the FEZ-1 metallo-β-lactamaseLiénard, Benoît M.R. / Horsfall, Louise E. / Galleni, Moreno / Frère, Jean-Marie / Schofield, Christopher J. et al. | 2006
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13C bis-labeled pyrroles: A tool for the identification of the rat metabolism of 3-methyl pyrrole-2,4-dicarboxylic acid 2-propyl ester 4-(1,2,2-trimethyl-propyl) esterMicheli, Fabrizio / Cavanni, Paolo / Fabio, Romano Di / Donati, Daniele / Hamdan, Mahmoud / Provera, Stefano / Tranquillini, Maria Elvira / Vitulli, Giovanni et al. | 2006
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Novel 1H-(benzimidazol-2-yl)-1H-pyridin-2-one inhibitors of insulin-like growth factor I (IGF-1R) kinaseWittman, Mark D. / Balasubramanian, Balu / Stoffan, Karen / Velaparthi, Upender / Liu, Pieying / Krishnanathan, Subramaniam / Carboni, Joan / Li, Aixin / Greer, Ann / Attar, Ricardo et al. | 2006
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Efficient synthesis of substituted 7-methyl-2H,5H-pyrano[4,3-b]pyran-5-ones and evaluation of their in vitro antiproliferative/cytotoxic activitiesLeutbecher, Heiko / Williams, Lawrence A.D. / Rösner, Harald / Beifuss, Uwe et al. | 2006
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Synthesis and biological evaluation of the suberoylanilide hydroxamic acid (SAHA) b-glucuronide and b-galactoside for application in selective prodrug chemotherapyThomas, M. / Rivault, F. / Tranoy-Opalinski, I. / Roche, J. / Gesson, J. P. / Papot, S. et al. | 2007
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Inhibition of membrane-associated carbonic anhydrase isozymes IX, XII and XIV with a library of glycoconjugate benzenesulfonamidesWilkinson, Brendan L. / Bornaghi, Laurent F. / Houston, Todd A. / Innocenti, Alessio / Vullo, Daniela / Supuran, Claudiu T. / Poulsen, Sally-Ann et al. | 2006
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Discovery of (Z)-2-phenyl-3-(1H-pyrrol-2-yl)acrylonitrile derivatives active against Haemonchus contortus and Ctenocephalides felis (cat flea)Ali, Abdelselam / Bliese, Marianne / Rasmussen, Jo-Anne M. / Sargent, Roger M. / Saubern, Simon / Sawutz, David G. / Wilkie, John S. / Winkler, David A. / Winzenberg, Kevin N. / Woodgate, Ruth C.J. et al. | 2006
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Editorial board| 2007
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Instructions to contributors| 2007