Synthesis and in vitro anti-proliferative activity of β-elemene monosubstituted derivatives in HeLa cells mediated through arrest of cell cycle at the G1 phase (English)
- New search for: Sun, Yanhong
- New search for: Sun, Yanhong
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In:
Bioorganic & medicinal chemistry
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17
, 3
; 1118-1124
;
2009
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ISSN:
- Article (Journal) / Print
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Title:Synthesis and in vitro anti-proliferative activity of β-elemene monosubstituted derivatives in HeLa cells mediated through arrest of cell cycle at the G1 phase
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Contributors:
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Published in:Bioorganic & medicinal chemistry ; 17, 3 ; 1118-1124
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Publisher:
- New search for: Elsevier
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Place of publication:Amsterdam [u.a.]
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Publication date:2009
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ISSN:
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ZDBID:
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Type of media:Article (Journal)
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Type of material:Print
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Language:English
- New search for: 35.70 / 44.33 / 44.40
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Source:
Table of contents – Volume 17, Issue 3
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 935
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Graphical contents list| 2009
- 950
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Tetrahedron Young Investigator Award for Bioorganic and Medicinal ChemistryWong, Chi-Huey et al. | 2009
- 951
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Biographical Sketch: Professor Jonathan Ellman| 2009
- 952
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b-Turn secondary structure and melanocortin ligandsHaslach, E. M. / Schaub, J. W. / Haskell-Luevano, C. et al. | 2009
- 952
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β-Turn secondary structure and melanocortin ligandsHaslach, Erica M. / Schaub, Jay W. / Haskell-Luevano, Carrie et al. | 2008
- 959
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Synthesis, penetrability and intracellular targeting of fluorescein-tagged peptoids and peptide–peptoid hybridsUnciti-Broceta, Asier / Diezmann, Franziska / Ou-Yang, Chiung Ying / Fara, Mario Antonio / Bradley, Mark et al. | 2008
- 967
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Sidechain-linked inhibitors of HIV-1 protease dimerizationBowman, Michael J. / Chmielewski, Jean et al. | 2008
- 977
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A small molecule inhibitor of a4 integrin-dependent cell migrationLee, J. / Hong, J. / Nam, T. G. / Peters, E. C. / Orth, A. P. / Geierstanger, B. H. / Goldfinger, L. E. / Ginsberg, M. H. / Cho, C. Y. / Schultz, P. G. et al. | 2009
- 977
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A small molecule inhibitor of α4 integrin-dependent cell migrationLee, Jongkook / Hong, Jiyong / Nam, Tae-Gyu / Peters, Eric C. / Orth, Anthony P. / Geierstanger, Bernhard H. / Goldfinger, Lawrence E. / Ginsberg, Mark H. / Cho, Charles Y. / Schultz, Peter G. et al. | 2008
- 981
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Site-specific covalent labeling of proteins inside live cells using small molecule probesChattopadhaya, Souvik / Srinivasan, Rajavel / Yeo, Dawn S.Y. / Chen, Grace Y.J. / Yao, Shao Q. et al. | 2008
- 990
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High throughput screening of potentially selective MMP-13 exosite inhibitors utilizing a triple-helical FRET substrateLauer-Fields, Janelle L. / Minond, Dmitriy / Chase, Peter S. / Baillargeon, Pierre E. / Saldanha, S. Adrian / Stawikowska, Roma / Hodder, Peter / Fields, Gregg B. et al. | 2008
- 1006
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Synthesis and preliminary antibacterial evaluation of simplified thiomarinol analogsMarion, Olivier / Gao, Xuri / Marcus, Sandra / Hall, Dennis G. et al. | 2008
- 1018
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On-bead cyclization in a combinatorial library of 15,625 octapeptidesFluxa, Viviana S. / Reymond, Jean-Louis et al. | 2008
- 1026
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Synthesis and screening of a cyclic peptide library: Discovery of small-molecule ligands against human prolactin receptorLiu, Tao / Joo, Sang Hoon / Voorhees, Jeffrey L. / Brooks, Charles L. / Pei, Dehua et al. | 2008
- 1034
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Expanding the repertoire of small molecule transcriptional activation domainsCasey, Ryan J. / Desaulniers, Jean-Paul / Hojfeldt, Jonas W. / Mapp, Anna K. et al. | 2008
- 1044
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Synthesis and biological evaluation of a library of resveratrol analogues as inhibitors of COX-1, COX-2 and NF-kBKang, S. S. / Cuendet, M. / Endringer, D. C. / Croy, V. L. / Pezzuto, J. M. / Lipton, M. A. et al. | 2009
- 1044
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Synthesis and biological evaluation of a library of resveratrol analogues as inhibitors of COX-1, COX-2 and NF-κBKang, Soo Sung / Cuendet, Muriel / Endringer, Denise C. / Croy, Vicki L. / Pezzuto, John M. / Lipton, Mark A. et al. | 2008
- 1055
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Coulombic effects on the traceless Staudinger ligation in waterTam, Annie / Raines, Ronald T. et al. | 2008
- 1064
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Substrate optimization for monitoring cathepsin C activity in live cellsLi, Jun / Petrassi, H. Michael / Tumanut, Christine / Masick, Brian T. / Trussell, Christopher / Harris, Jennifer L. et al. | 2008
- 1071
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Evaluation of α,β-unsaturated ketone-based probes for papain-family cysteine proteasesYang, Zhimou / Fonović, Marko / Verhelst, Steven H.L. / Blum, Galia / Bogyo, Matthew et al. | 2008
- 1071
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Evaluation of a,b-unsaturated ketone-based probes for papain-family cysteine proteasesYang, Z. / Fonovic, M. / Verhelst, S. H. / Blum, G. / Bogyo, M. et al. | 2009
- 1079
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ATP competitive inhibitors of d-alanine–d-alanine ligase based on protein kinase inhibitor scaffoldsTriola, Gemma / Wetzel, Stefan / Ellinger, Bernhard / Koch, Marcus A. / Hübel, Katja / Rauh, Daniel / Waldmann, Herbert et al. | 2008
- 1088
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A road less traveled by: Exploring a decade of Ellman chemistryShelat, Anang A. / Guy, R. Kiplin et al. | 2008
- 1094
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Using specificity to strategically target proteasesLim, Mark D. / Craik, Charles S. et al. | 2008
- 1101
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Ranking the selectivity of PubChem screening hits by activity-based protein profiling: MMP13 as a case studyNakai, Ryuichiro / Salisbury, Cleo M. / Rosen, Hugh / Cravatt, Benjamin F. et al. | 2008
- 1109
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Synthesis and biological evaluation of p-carborane bisphenols and their derivatives: Structure–activity relationship for estrogenic activityOgawa, Takumi / Ohta, Kiminori / Iijima, Toru / Suzuki, Tomoharu / Ohta, Shigeru / Endo, Yasuyuki et al. | 2008
- 1118
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Synthesis and in vitro anti-proliferative activity of β-elemene monosubstituted derivatives in HeLa cells mediated through arrest of cell cycle at the G1 phaseSun, Yanhong / Liu, Guifeng / Zhang, Yuangqing / Zhu, Hua / Ren, Yunfeng / Shen, Yu-Mei et al. | 2008
- 1118
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Synthesis and in vitro anti-proliferative activity of b-elemene monosubstituted derivatives in HeLa cells mediated through arrest of cell cycle at the G1 phaseSun, Y. / Liu, G. / Zhang, Y. / Zhu, H. / Ren, Y. / Shen, Y. M. et al. | 2009
- 1125
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Novel 6-methanesulfonamide-3,4-methylenedioxyphenyl-N-acylhydrazones: Orally effective anti-inflammatory drug candidatesTributino, Jorge L.M. / Duarte, Carolina D. / Corrêa, Rodrigo S. / Doriguetto, Antonio C. / Ellena, Javier / Romeiro, Nelilma C. / Castro, Newton G. / Miranda, Ana Luisa P. / Barreiro, Eliezer J. / Fraga, Carlos A.M. et al. | 2008
- 1132
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Benzopyridooxathiazepine derivatives as novel potent antimitotic agentsGallet, Sebastien / Flouquet, Nathalie / Carato, Pascal / Pfeiffer, Bruno / Renard, Pierre / Léonce, Stéphane / Pierré, Alain / Berthelot, Pascal / Lebegue, Nicolas et al. | 2008
- 1139
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Solution- and solid-phase synthesis and anti-HIV activity of maslinic acid derivatives containing amino acids and peptidesParra, Andres / Rivas, Francisco / Lopez, Pilar E. / Garcia-Granados, Andres / Martinez, Antonio / Albericio, Fernando / Marquez, Nieves / Muñoz, Eduardo et al. | 2008
- 1146
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Synthesis and cyclooxygenase inhibition of various (aryl-1,2,3-triazole-1-yl)-methanesulfonylphenyl derivativesWuest, Frank / Tang, Xinli / Kniess, Torsten / Pietzsch, Jens / Suresh, Mavanur et al. | 2008
- 1152
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Function-oriented synthesis applied to the anti-botulinum natural product toosendaninNakai, Yuya / Tepp, William H. / Dickerson, Tobin J. / Johnson, Eric A. / Janda, Kim D. et al. | 2008
- 1158
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Carbonic anhydrase inhibitors: Inhibition of the β-class enzyme from the yeast Saccharomyces cerevisiae with sulfonamides and sulfamatesIsik, Semra / Kockar, Feray / Aydin, Meltem / Arslan, Oktay / Guler, Ozen Ozensoy / Innocenti, Alessio / Scozzafava, Andrea / Supuran, Claudiu T. et al. | 2008
- 1158
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Carbonic anhydrase inhibitors: Inhibition of the b-class enzyme from the yeast Saccharomyces cerevisiae with sulfonamides and sulfamatesIsik, S. / Kockar, F. / Aydin, M. / Arslan, O. / Guler, O. O. / Innocenti, A. / Scozzafava, A. / Supuran, C. T. et al. | 2009
- 1164
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In vitro solubility, stability and permeability of novel quercetin–amino acid conjugatesKim, Mi Kyoung / Park, Kwang-su / Yeo, Woon-seok / Choo, Hyunah / Chong, Youhoon et al. | 2008
- 1172
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Synthesis and antitumor activity of novel enediyne-linked pyrrolo[2,1-c][1,4]benzodiazepine hybridsHu, Wan-Ping / Liang, Jium-Jia / Kao, Chai-Lin / Chen, You-Chiang / Chen, Chung-Yu / Tsai, Feng-Yuan / Wu, Ming-Jung / Chang, Long-Sen / Chen, Yeh-Long / Wang, Jeh-Jeng et al. | 2008
- 1181
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Death receptor 5 targeting activity-guided isolation of isoflavones from Millettia brandisiana and Ardisia colorata and evaluation of ability to induce TRAIL-mediated apoptosisKikuchi, Hiroyuki / Ohtsuki, Takashi / Koyano, Takashi / Kowithayakorn, Thaworn / Sakai, Toshiyuki / Ishibashi, Masami et al. | 2008
- 1187
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Synthesis of buprestins D, E, F, G and H; structural confirmation and biological testing of acyl glucoses from jewel beetles (Coleoptera: Buprestidae)Ryczek, Sebastian / Dettner, Konrad / Unverzagt, Carlo et al. | 2008
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Discovery of N-[(1R,2S,5S)-2-{[(5-chloroindol-2-yl)carbonyl]amino}-5-(dimethylcarbamoyl)cyclohexyl]-5-methyl-4,5,6,7-tetrahydrothiazolo[5,4-c]pyridine-2-carboxamide hydrochloride: A novel, potent and orally active direct inhibitor of factor XaNagata, Tsutomu / Yoshino, Toshiharu / Haginoya, Noriyasu / Yoshikawa, Kenji / Nagamochi, Masatoshi / Kobayashi, Syozo / Komoriya, Satoshi / Yokomizo, Aki / Muto, Ryo / Yamaguchi, Mitsuhiro et al. | 2008
- 1207
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Synthesis, structure and antibacterial activity of new 2-(1-(2-(substituted-phenyl)-5-methyloxazol-4-yl)-3-(2-substitued-phenyl)-4,5-dihydro-1H-pyrazol-5-yl)-7-substitued-1,2,3,4-tetrahydroisoquinoline derivativesLiu, Xin-Hua / Zhu, Jing / Zhou, An-na / Song, Bao-An / Zhu, Hai-Liang / bai, Lin-Shan / Bhadury, Pinaki S. / Pan, Chun-Xiu et al. | 2008
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Carbonic anhydrase inhibitors. Comparison of chlorthalidone, indapamide, trichloromethiazide, and furosemide X-ray crystal structures in adducts with isozyme II, when several water molecules make the differenceTemperini, Claudia / Cecchi, Alessandro / Scozzafava, Andrea / Supuran, Claudiu T. et al. | 2008
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New N-substituted 9-azabicyclo[3.3.1]nonan-3α-yl phenylcarbamate analogs as σ2 receptor ligands: Synthesis, in vitro characterization, and evaluation as PET imaging and chemosensitization agentsChu, Wenhua / Xu, Jinbin / Zhou, Dong / Zhang, Fanjie / Jones, Lynne A. / Wheeler, Kenneth T. / Mach, Robert H. et al. | 2008
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New N-substituted 9-azabicyclo[3.3.1]nonan-3a-yl phenylcarbamate analogs as 2 receptor ligands: Synthesis, in vitro characterization, and evaluation as PET imaging and chemosensitization agentsChu, W. / Xu, J. / Zhou, D. / Zhang, F. / Jones, L. A. / Wheeler, K. T. / Mach, R. H. et al. | 2009
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A novel and potent VLA-4 antagonist based on trans-4-substituted cyclohexanecarboxylic acidMuro, Fumihito / Iimura, Shin / Yoneda, Yoshiyuki / Chiba, Jun / Watanabe, Toshiyuki / Setoguchi, Masaki / Takayama, Gensuke / Yokoyama, Mika / Takashi, Tohru / Nakayama, Atsushi et al. | 2008
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Correlation of binding constants and molecular modelling of inhibitors in the active sites of aldose reductase and aldehyde reductaseCarbone, Vincenzo / Zhao, Hai-Tao / Chung, Roland / Endo, Satoshi / Hara, Akira / El-Kabbani, Ossama et al. | 2008
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Conformational analysis of trimeric maleimide substituted 1,5,9-triazacyclododecane HIV fusion scaffoldsRemmert, Sarah / Hollis, Heather / Parish, Carol A. et al. | 2008
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Structure–activity relationship study on polyglutamine binding peptide QBP1Tomita, Kenji / Popiel, H. Akiko / Nagai, Yoshitaka / Toda, Tatsushi / Yoshimitsu, Yuji / Ohno, Hiroaki / Oishi, Shinya / Fujii, Nobutaka et al. | 2008
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Novel DNA-directed alkylating agents: Design, synthesis and potent antitumor effect of phenyl N-mustard-9-anilinoacridine conjugates via a carbamate or carbonate linkerKapuriya, Naval / Kapuriya, Kalpana / Dong, Huajin / Zhang, Xiuguo / Chou, Ting-Chao / Chen, Yu-Ting / Lee, Te-Chang / Lee, Wen-Chuan / Tsai, Tung-Hu / Naliapara, Yogesh et al. | 2008
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Towards Gram-negative antivirulence drugs: New inhibitors of HldE kinaseDesroy, Nicolas / Moreau, François / Briet, Sophia / Fralliec, Géraldine Le / Floquet, Stephanie / Durant, Lionel / Vongsouthi, Vanida / Gerusz, Vincent / Denis, Alexis / Escaich, Sonia et al. | 2008
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Synthesis and biological evaluation of curcuminoid pyrazoles as new therapeutic agents in inflammatory bowel disease: Effect on matrix metalloproteinasesClaramunt, R.M. / Bouissane, L. / Cabildo, M.P. / Cornago, M.P. / Elguero, J. / Radziwon, A. / Medina, C. et al. | 2008
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Solid-phase parallel synthesis and SAR of 4-amidofuran-3-one inhibitors of cathepsin S: Effect of sulfonamides P3 substituents on potency and selectivityAyesa, Susana / Lindquist, Charlotta / Agback, Tatiana / Benkestock, Kurt / Classon, Björn / Henderson, Ian / Hewitt, Ellen / Jansson, Katarina / Kallin, Anders / Sheppard, Dave et al. | 2008
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Instructions to contributors| 2009
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Editorial board| 2009