Modified tetrahalogenated benzimidazoles with CK2 inhibitory activity are active against human prostate cancer cells LNCaP in vitro (English)
- New search for: Schneider, Carolin C.
- New search for: Schneider, Carolin C.
- New search for: Kartarius, Sabine
- New search for: Montenarh, Mathias
- New search for: Orzeszko, Andrzej
- New search for: Kazimierczuk, Zygmunt
In:
Bioorganic & medicinal chemistry
;
20
, 14
; 4390-4397
;
2012
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ISSN:
- Article (Journal) / Print
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Title:Modified tetrahalogenated benzimidazoles with CK2 inhibitory activity are active against human prostate cancer cells LNCaP in vitro
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Contributors:
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Published in:Bioorganic & medicinal chemistry ; 20, 14 ; 4390-4397
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Publisher:
- New search for: Elsevier
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Place of publication:Amsterdam [u.a.]
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Publication date:2012
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ISSN:
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ZDBID:
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Type of media:Article (Journal)
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Type of material:Print
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Language:English
- New search for: 35.70 / 44.33 / 44.40
- Further information on Basic classification
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Keywords:
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Source:
Table of contents – Volume 20, Issue 14
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 4173
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Graphical contents list| 2012
- 4186
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The effect on quadruplex stability of North-nucleoside derivatives in the loops of the thrombin-binding aptamerAviñó, Anna / Mazzini, Stefania / Ferreira, Ruben / Gargallo, Raimundo / Marquez, Victor E. / Eritja, Ramon et al. | 2012
- 4194
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Structure-based design of rhodanine-based acylsulfonamide derivatives as antagonists of the anti-apoptotic Bcl-2 proteinLi, Huan-qiu / Yang, Jing / Ma, Shuhua / Qiao, Chunhua et al. | 2012
- 4201
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Novel retinoic acid 4-hydroxylase (CYP26) inhibitors based on a 3-(1H-imidazol- and triazol-1-yl)-2,2-dimethyl-3-(4-(phenylamino)phenyl)propyl scaffoldGomaa, Mohamed S. / Bridgens, Caroline E. / Illingworth, Nicola A. / Veal, Gareth J. / Redfern, Christopher P.F. / Brancale, Andrea / Armstrong, Jane L. / Simons, Claire et al. | 2012
- 4208
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Design, synthesis and biological activity of 6-substituted carbamoyl benzimidazoles as new nonpeptidic angiotensin II AT1 receptor antagonistsZhang, Jun / Wang, Jin-Liang / Zhou, Zhi-Ming / Li, Zhi-Huai / Xue, Wei-Zhe / Xu, Di / Hao, Li-Ping / Han, Xiao-Feng / Fei, Fan / Liu, Ting et al. | 2012
- 4217
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Novel tricyclic indeno[2,1-d]pyrimidines with dual antiangiogenic and cytotoxic activities as potent antitumor agentsGangjee, Aleem / Zhao, Ying / Ihnat, Michael A. / Thorpe, Jessica E. / Bailey-Downs, Lora C. / Kisliuk, Roy L. et al. | 2012
- 4226
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Design, synthesis, biological evaluation and molecular modeling of novel 1,3,4-oxadiazole derivatives based on Vanillic acid as potential immunosuppressive agentsTang, Jian-Feng / Lv, Xian-Hai / Wang, Xiao-Liang / Sun, Jian / Zhang, Yan-Bin / Yang, Yu-Shun / Gong, Hai-Bin / Zhu, Hai-Liang et al. | 2012
- 4237
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Novel 5-substituted benzyloxy-2-arylbenzofuran-3-carboxylic acids as calcium activated chloride channel inhibitorsKumar, Satish / Namkung, Wan / Verkman, A.S. / Sharma, Pawan K. et al. | 2012
- 4245
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Synthesis and SAR-study for novel arylpiperazine derivatives of 5-arylidenehydantoin with a1-adrenoceptor antagonistic propertiesHandzlik, J. / Szymanska, E. / Wojcik, R. / Dela, A. / Jastrzebska-Wiesek, M. / Karolak-Wojciechowska, J. / Fruzinski, A. / Siwek, A. / Filipek, B. / Kiec-Kononowicz, K. et al. | 2012
- 4245
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Synthesis and SAR-study for novel arylpiperazine derivatives of 5-arylidenehydantoin with α1-adrenoceptor antagonistic propertiesHandzlik, Jadwiga / Szymańska, Ewa / Wójcik, Renata / Dela, Anna / Jastrzębska-Więsek, Magdalena / Karolak-Wojciechowska, Janina / Fruziński, Andrzej / Siwek, Agata / Filipek, Barbara / Kieć-Kononowicz, Katarzyna et al. | 2012
- 4258
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- 4271
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Synthesis and biological evaluation of novel anticancer bivalent colchicine–tubulizine hybridsMalysheva, Yulia B. / Combes, Sebastien / Allegro, Diane / Peyrot, Vincent / Knochel, Paul / Gavryushin, Andrei E. / Fedorov, Alexey Yu. et al. | 2012
- 4279
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Synthesis and structure–activity relationships of benzophenone-bearing diketopiperazine-type anti-microtubule agentsYamazaki, Yuri / Sumikura, Makiko / Masuda, Yurika / Hayashi, Yoshiki / Yasui, Hiroyuki / Kiso, Yoshiaki / Chinen, Takumi / Usui, Takeo / Yakushiji, Fumika / Potts, Barbara et al. | 2012
- 4290
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Thiorhodamines containing amide and thioamide functionality as inhibitors of the ATP-binding cassette drug transporter P-glycoprotein (ABCB1)Orchard, Alexandra / Schamerhorn, Gregory A. / Calitree, Brandon D. / Sawada, Geri A. / Loo, Tip W. / Claire Bartlett, M. / Clarke, David M. / Detty, Michael R. et al. | 2012
- 4303
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Bisubstrate analog inhibitors of 6-hydroxymethyl-7,8-dihydropterin pyrophosphokinase: New lead exhibits a distinct binding modeShi, Genbin / Shaw, Gary / Li, Yue / Wu, Yan / Yan, Honggao / Ji, Xinhua et al. | 2012
- 4310
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Quencher-free molecular beacon tethering 7-hydroxycoumarin detects targets through protonation/deprotonationKashida, Hiromu / Yamaguchi, Kyohei / Hara, Yuichi / Asanuma, Hiroyuki et al. | 2012
- 4316
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- 4323
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Design, synthesis and antitumor activities of novel bis-aryl ureas derivatives as Raf kinase inhibitorsZhan, Wenhu / Li, Yanyang / Huang, Weiping / Zhao, Yanjin / Yao, Zhenglin / Yu, Shanyou / Yuan, Shoujun / Jiang, Falong / Yao, Shan / Li, Shuxin et al. | 2012
- 4330
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Synthesis and evaluation of a radioiodinated bladder cancer specific peptideHa, Yeong Su / Lee, Hwa Young / An, Gwang Il / Kim, Jonghee / Kwak, Wonjung / Lee, Eun-Ju / Lee, Seung-Min / Lee, Byung-Heon / Kim, In-San / Belay, Takele et al. | 2012
- 4336
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Inhibition of monoamine oxidase by 8-phenoxymethylcaffeine derivativesOkaecwe, Thokozile / Swanepoel, Abraham J. / Petzer, Anél / Bergh, Jacobus J. / Petzer, Jacobus P. et al. | 2012
- 4348
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Myxobacteria versus sponge-derived alkaloids: The bengamide family identified as potent immune modulating agents by scrutiny of LC–MS/ELSD librariesJohnson, Tyler A. / Sohn, Johann / Vaske, Yvette M. / White, Kimberly N. / Cohen, Tanya L. / Vervoort, Helene C. / Tenney, Karen / Valeriote, Frederick A. / Bjeldanes, Leonard F. / Crews, Phillip et al. | 2012
- 4356
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Functional characterization of recombinant hyoscyamine 6b-hydroxylase from Atropa belladonnaLi, J. / van Belkum, M. J. / Vederas, J. C. et al. | 2012
- 4356
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Functional characterization of recombinant hyoscyamine 6β-hydroxylase from Atropa belladonnaLi, Jing / van Belkum, Marco J. / Vederas, John C. et al. | 2012
- 4364
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- 4371
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- 4390
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Modified tetrahalogenated benzimidazoles with CK2 inhibitory activity are active against human prostate cancer cells LNCaP in vitroSchneider, Carolin C. / Kartarius, Sabine / Montenarh, Mathias / Orzeszko, Andrzej / Kazimierczuk, Zygmunt et al. | 2012
- 4397
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Synthesis, biological evaluation and molecular docking studies of 3-(1,3-diphenyl-1H-pyrazol-4-yl)-N-phenylacrylamide derivatives as inhibitors of HDAC activityLi, Xi / Liu, Jia-Lin / Yang, Xian-Hui / Lu, Xiang / Zhao, Ting-Ting / Gong, Hai-Bin / Zhu, Hai-Liang et al. | 2012
- 4437
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- IFC
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Editorial board| 2012