1,2,3-Triazolyl-4-oxoquinolines: A feasible beginning for promising chemical structures to inhibit oseltamivir-resistant influenza A and B viruses (English)
- New search for: Boechat, Fernanda da C S
- New search for: Boechat, Fernanda da C S
- New search for: Sacramento, Carolina Q
- New search for: Cunha, Anna C
- New search for: Sagrillo, Fernanda S
- New search for: Nogueira, Christiane M
- New search for: Fintelman-Rodrigues, Natalia
- New search for: Santos-Filho, Osvaldo
- New search for: Riscado, Cecília S
- New search for: Forezi, Luana da S M
- New search for: Faro, Letícia V
- New search for: Brozeguini, Leonardo
- New search for: Marques, Isakelly P
- New search for: Ferreira, Vitor F
- New search for: Souza, Thiago Moreno L
- New search for: de Souza, Maria Cecília B V
In:
Bioorganic & medicinal chemistry
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23
, 24
; 7777-7784
;
2015
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ISSN:
- Article (Journal) / Print
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Title:1,2,3-Triazolyl-4-oxoquinolines: A feasible beginning for promising chemical structures to inhibit oseltamivir-resistant influenza A and B viruses
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Contributors:
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Published in:Bioorganic & medicinal chemistry ; 23, 24 ; 7777-7784
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Publisher:
- New search for: Elsevier
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Place of publication:Amsterdam [u.a.]
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Publication date:2015
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ISSN:
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ZDBID:
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DOI:
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Type of media:Article (Journal)
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Type of material:Print
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Language:English
- New search for: 35.70 / 44.33 / 44.40
- Further information on Basic classification
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Keywords:
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Source:
Table of contents – Volume 23, Issue 24
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 7489
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Graphical contents list| 2015
- 7497
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Structural interrogation of benzosuberene-based inhibitors of tubulin polymerizationHerdman, Christine A. / Devkota, Laxman / Lin, Chen-Ming / Niu, Haichan / Strecker, Tracy E. / Lopez, Ramona / Liu, Li / George, Clinton S. / Tanpure, Rajendra P. / Hamel, Ernest et al. | 2015
- 7521
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Synthesis and evaluation of 3-hydroxy-3-phenylpropanoate ester–AZT conjugates as potential dual-action HIV-1 Integrase and Reverse Transcriptase inhibitorsManyeruke, Meloddy H. / Olomola, Temitope O. / Majumder, Swarup / Abrahams, Shaakira / Isaacs, Michelle / Mautsa, Nicodemus / Mosebi, Salerwe / Mnkandhla, Dumisani / Hewer, Raymond / Hoppe, Heinrich C. et al. | 2015
- 7529
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Synthesis and comparison of the biological activity of monocyclic phosphonate, difluorophosphonate and phosphate analogs of the natural AChE inhibitor cyclophostinMartin, Benjamin P. / Vasilieva, Elena / Dupureur, Cynthia M. / Spilling, Christopher D. et al. | 2015
- 7535
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Synthesis and activity of novel 16-dehydropregnenolone acetate derivatives as inhibitors of type 1 5α-reductase and on cancer cell line SK-LU-1Silva-Ortiz, Aylin Viviana / Bratoeff, Eugene / Ramírez-Apan, Teresa / Heuze, Yvonne / Sánchez, Araceli / Soriano, Juan / Cabeza, Marisa et al. | 2015
- 7543
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A structure–activity relationship of non-peptide macrocyclic histone deacetylase inhibitors and their anti-proliferative and anti-inflammatory activitiesTapadar, Subhasish / Fathi, Shaghayegh / Raji, Idris / Omesiete, Wilson / Kornacki, James R. / Mwakwari, Sandra C. / Miyata, Masanori / Mitsutake, Kazunori / Li, Jian-Dong / Mrksich, Milan et al. | 2015
- 7565
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Targeting quorum sensing by designing azoline derivatives to inhibit the N-hexanoyl homoserine lactone-receptor CviR: Synthesis as well as biological and theoretical evaluationsBucio-Cano, Alejandro / Reyes-Arellano, Alicia / Correa-Basurto, José / Bello, Martiniano / Torres-Jaramillo, Jenifer / Salgado-Zamora, Héctor / Curiel-Quesada, Everardo / Peralta-Cruz, Javier / Avila-Sorrosa, Alcives et al. | 2015
- 7578
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Localization-dependent cell-killing effects of protoporphyrin (PPIX)-lipid micelles and liposomes in photodynamic therapyTachikawa, Shoji / Sato, Shinichi / Hazama, Hisanao / Kaneda, Yasufumi / Awazu, Kunio / Nakamura, Hiroyuki et al. | 2015
- 7585
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Discovery of novel quinoline-based mTOR inhibitors via introducing intra-molecular hydrogen bonding scaffold (iMHBS): The design, synthesis and biological evaluationMa, Xiaodong / Lv, Xiaoqing / Qiu, Ni / Yang, Bo / He, Qiaojun / Hu, Yongzhou et al. | 2015
- 7597
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Design, synthesis and evaluation of antiestrogen and histone deacetylase inhibitor molecular hybridsMendoza-Sanchez, Rodrigo / Cotnoir-White, David / Kulpa, Justyna / Jutras, Isabel / Pottel, Joshua / Moitessier, Nicolas / Mader, Sylvie / Gleason, James L. et al. | 2015
- 7607
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Searching for novel applications of the benzohomoadamantane scaffold in medicinal chemistry: Synthesis of novel 11β-HSD1 inhibitorsValverde, Elena / Seira, Constantí / McBride, Andrew / Binnie, Margaret / Luque, F. Javier / Webster, Scott P. / Bidon-Chanal, Axel / Vázquez, Santiago et al. | 2015
- 7618
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Synthesis, antiviral activity and resistance of a novel small molecule HIV-1 entry inhibitorCurreli, Francesca / Haque, Kashfia / Xie, Lihua / Qiu, Qian / Xu, Jinfeng / Yong, Weizhong / Tong, Xiaohe / Debnath, Asim K. et al. | 2015
- 7629
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Synthesis and bio-evaluation of novel quinolino-stilbene derivatives as potential anticancer agentsSrivastava, Vandana / Lee, Hoyun et al. | 2015
- 7641
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Phenolic group on A-ring is key for dracoflavan B as a selective noncompetitive inhibitor of α-amylaseToh, Zhi Siang / Wang, Hongyu / Yip, Yew Mun / Lu, Yuyun / Lim, Benedict Jeffrey Ang / Zhang, Daiwei / Huang, Dejian et al. | 2015
- 7650
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Modification of a dihydropyrrolopyrimidine phosphoinositide 3-kinase (PI3K) inhibitor to improve oral bioavailabilityKawada, Hatsuo / Ebiike, Hirosato / Tsukazaki, Masao / Yamamoto, Shun / Koyama, Kohei / Nakamura, Mitsuaki / Morikami, Kenji / Yoshinari, Kiyoshi / Yoshida, Miyuki / Ogawa, Kotaro et al. | 2015
- 7661
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Small molecules enhance functional O-mannosylation of Alpha-dystroglycanLv, Fengping / Li, Zhi-fang / Hu, Wenhao / Wu, Xiaohua et al. | 2015
- 7671
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Singlet oxygen oxidation products of biliverdin IXα dimethyl esterDorazio, Sarina J. / Halepas, Steven / Bruhn, Torsten / Fleming, Kathleen M. / Zeller, Matthias / Brückner, Christian et al. | 2015
- 7676
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Identification of dual PPARα/γ agonists and their effects on lipid metabolismGao, Quanqing / Hanh, Jacky / Váradi, Linda / Cairns, Rose / Sjöström, Helena / Liao, Vivian W.Y. / Wood, Peta / Balaban, Seher / Ong, Jennifer Ai / Lin, Hsuan-Yu Jennifer et al. | 2015
- 7685
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Design, synthesis and preliminary biological studies of pyrrolidine derivatives as Mcl-1 inhibitorsWan, Yichao / Wang, Junhua / Sun, Feng’e / Chen, Minglu / Hou, Xuben / Fang, Hao et al. | 2015
- 7694
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Discovery of benzothiazoles as antimycobacterial agents: Synthesis, structure–activity relationships and binding studies with Mycobacterium tuberculosis decaprenylphosphoryl-β-d-ribose 2′-oxidaseLandge, Sudhir / Mullick, Amrita B. / Nagalapur, Kavitha / Neres, João / Subbulakshmi, Venkita / Murugan, Kannan / Ghosh, Anirban / Sadler, Claire / Fellows, Mick D. / Humnabadkar, Vaishali et al. | 2015
- 7711
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Pyrazole clubbed triazolo[1,5-a]pyrimidine hybrids as an anti-tubercular agents: Synthesis, in vitro screening and molecular docking studyBhatt, Jaimin D. / Chudasama, Chaitanya J. / Patel, Kanuprasad D. et al. | 2015
- 7717
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Discovery of 2-aryloxy-4-amino-quinazoline derivatives as novel protease-activated receptor 2 (PAR2) antagonistsCho, Nam-Chul / Cha, Ji Hyoun / Kim, Hyojin / Kwak, Jinsook / Kim, Dohee / Seo, Seung-Hwan / Shin, Ji-Sun / Kim, TaeHun / Park, Ki Duk / Lee, Jiyoun et al. | 2015
- 7728
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(E)-2-Cyano-3-(substituted phenyl)acrylamide analogs as potent inhibitors of tyrosinase: A linear β-phenyl-α,β-unsaturated carbonyl scaffoldSon, Sujin / Kim, Haewon / Yun, Hwi Young / Kim, Do Hyun / Ullah, Sultan / Kim, Seong Jin / Kim, Yeon-Jeong / Kim, Min-Soo / Yoo, Jin-Wook / Chun, Pusoon et al. | 2015
- 7735
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Synthesis, structure–activity relationship and biological evaluation of novel arylpiperzines as α1A/1D-AR subselective antagonists for BPHXu, Fang / Chen, Hong / Xu, Jingyi / Liang, Xue / He, Xuelan / Shao, Binhao / Sun, Xianqiang / Li, Bing / Deng, Xiaoliang / Yuan, Mu et al. | 2015
- 7743
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Development of 68Ga-labeled multivalent nitroimidazole derivatives for hypoxia imagingSeelam, Sudhakara Reddy / Lee, Ji Youn / Lee, Yun-Sang / Hong, Mi Kyung / Kim, Young Joo / Banka, Vinay Kumar / Lee, Dong Soo / Chung, June-Key / Jeong, Jae Min et al. | 2015
- 7751
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Benzenesulfonamides incorporating bulky aromatic/heterocyclic tails with potent carbonic anhydrase inhibitory activityBozdag, Murat / Alafeefy, Ahmed M. / Vullo, Daniela / Carta, Fabrizio / Dedeoglu, Nurcan / Al-Tamimi, Abdul-Malek S. / Al-Jaber, Nabila A. / Scozzafava, Andrea / Supuran, Claudiu T. et al. | 2015
- 7765
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Synthesis and antitumor activity evaluation of PI3K inhibitors containing 3-substituted quinazolin-4(3H)-one moietyZhang, Hao / Xin, Min-Hang / Xie, Xiao-Xiao / Mao, Shuai / Zuo, Sai-Jie / Lu, She-Min / Zhang, San-Qi et al. | 2015
- 7777
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1,2,3-Triazolyl-4-oxoquinolines: A feasible beginning for promising chemical structures to inhibit oseltamivir-resistant influenza A and B virusesBoechat, Fernanda da C.S. / Sacramento, Carolina Q. / Cunha, Anna C. / Sagrillo, Fernanda S. / Nogueira, Christiane M. / Fintelman-Rodrigues, Natalia / Santos-Filho, Osvaldo / Riscado, Cecília S. / Forezi, Luana da S.M. / Faro, Letícia V. et al. | 2015
- 7785
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Corrigendum to “Inhibition of human topoisomerase I and II and anti-proliferative effects on MCF-7 cells by new titanocene complexes” [Bioorg. Med. Chem. 23 (2015) 7302–7312]Chimento, Adele / Saturnino, Carmela / Iacopetta, Domenico / Mazzotta, Rosaria / Caruso, Anna / Plutino, Maria Rosaria / Mariconda, Annaluisa / Ramunno, Anna / Sinicropi, Maria Stefania / Pezzi, Vincenzo et al. | 2015
- 7786
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Corrigendum to “2-Arylquinazolin-4(3H)-ones: A new class of α-glucosidase inhibitors” [Bioorg. Med. Chem. 23 (2015) 7417–7421]Javaid, Kulsoom / Saad, Syed Muhammad / Rasheed, Saima / Moin, Syed Tarique / Syed, Naima / Fatima, Itrat / Salar, Uzma / Khan, Khalid Mohammed / Perveen, Shahnaz / Choudhary, M. Iqbal et al. | 2015
- IFC
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Editorial board| 2015