Biocatalysis at Work: Applications in the Development of Sagopilone (English)
- New search for: Gottfried, Kathrin
- New search for: Gottfried, Kathrin
- New search for: Klar, Ulrich
- New search for: Platzek, Johannes
- New search for: Zorn, Ludwig
In:
ChemMedChem
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10
, 7
; 1240-1248
;
2015
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ISSN:
- Article (Journal) / Print
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Title:Biocatalysis at Work: Applications in the Development of Sagopilone
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Contributors:
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Published in:ChemMedChem ; 10, 7 ; 1240-1248
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Publisher:
- New search for: Wiley-VCH
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Place of publication:Weinheim
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Publication date:2015
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ISSN:
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ZDBID:
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DOI:
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Type of media:Article (Journal)
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Type of material:Print
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Language:English
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Keywords:
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Classification:
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Source:
Table of contents – Volume 10, Issue 7
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 1117
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Cover Picture: Freezing the Bioactive Conformation to Boost Potency: The Identification of BAY 85‐8501, a Selective and Potent Inhibitor of Human Neutrophil Elastase for Pulmonary Diseases (ChemMedChem 7/2015)von Nussbaum, Franz / Li, Volkhart M.‐J. / Allerheiligen, Swen / Anlauf, Sonja / Bärfacker, Lars / Bechem, Martin / Delbeck, Martina / Fitzgerald, Mary F. / Gerisch, Michael / Gielen‐Haertwig, Heike et al. | 2015
- 1117
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Cover Picture: Freezing the Bioactive Conformation to Boost Potency: The Identification of BAY85-8501, a Selective and Potent Inhibitor of Human Neutrophil Elastase for Pulmonary DiseasesFranz vonNussbaum et al. | 2015
- 1118
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Inside Cover: Synthesis, Chiral Separation, Absolute Configuration Assignment, and Biological Activity of Enantiomers of Retro-1 as Potent Inhibitors of Shiga ToxinHajer Abdelkafi et al. | 2015
- 1118
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Inside Cover: Synthesis, Chiral Separation, Absolute Configuration Assignment, and Biological Activity of Enantiomers of Retro‐1 as Potent Inhibitors of Shiga Toxin (ChemMedChem 7/2015)Abdelkafi, Hajer / Michau, Aurélien / Clerget, Alexandra / Buisson, David‐Alexandre / Johannes, Ludger / Gillet, Daniel / Barbier, Julien / Cintrat, Jean‐Christophe et al. | 2015
- 1119
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Graphical Abstract: ChemMedChem 7/2015| 2015
- 1119
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Abstracts| 2015
- 1128
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Spotlights on our sister journals: ChemMedChem 7/2015| 2015
- 1133
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Medicinal Chemists of the 21st Century—Who Are We and Where to Go?Nussbaumer, Peter et al. | 2015
- 1141
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Protein Flexibility in Drug Discovery: From Theory to ComputationBuonfiglio, Rosa / Recanatini, Maurizio / Masetti, Matteo et al. | 2015
- 1149
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Potent, Metabolically Stable 2‐Alkyl‐8‐(2H‐1,2,3‐triazol‐2‐yl)‐9H‐adenines as Adenosine A2A Receptor LigandsPace, Silvia / Brogin, Giandomenico / Stasi, Maria Antonietta / Riccioni, Teresa / Borsini, Franco / Capocasa, Francesca / Manera, Francesco / Tallarico, Carlo / Grossi, Pietro / Vacondio, Federica et al. | 2015
- 1153
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Synthesis, Chiral Separation, Absolute Configuration Assignment, and Biological Activity of Enantiomers of Retro‐1 as Potent Inhibitors of Shiga ToxinAbdelkafi, Hajer / Michau, Aurélien / Clerget, Alexandra / Buisson, David‐Alexandre / Johannes, Ludger / Gillet, Daniel / Barbier, Julien / Cintrat, Jean‐Christophe et al. | 2015
- 1157
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A Phytochemical–Halogenated Quinoline Combination Therapy Strategy for the Treatment of Pathogenic BacteriaAbouelhassan, Yasmeen / Garrison, Aaron T. / Bai, Fang / Norwood, Verrill M. IV / Nguyen, Minh Thu / Jin, Shouguang / Huigens, Robert W. III et al. | 2015
- 1163
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Freezing the Bioactive Conformation to Boost Potency: The Identification of BAY 85‐8501, a Selective and Potent Inhibitor of Human Neutrophil Elastase for Pulmonary Diseasesvon Nussbaum, Franz / Li, Volkhart M.‐J. / Allerheiligen, Swen / Anlauf, Sonja / Bärfacker, Lars / Bechem, Martin / Delbeck, Martina / Fitzgerald, Mary F. / Gerisch, Michael / Gielen‐Haertwig, Heike et al. | 2015
- 1174
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Metabolic Instability of Cyanothiazolidine‐Based Prolyl Oligopeptidase Inhibitors: a Structural Assignment Challenge and Potential Medicinal Chemistry ImplicationsSchiavini, Paolo / Pottel, Joshua / Moitessier, Nicolas / Auclair, Karine et al. | 2015
- 1184
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Design, Synthesis, and Biological Evaluation of Novel Nonsteroidal Farnesoid X Receptor (FXR) Antagonists: Molecular Basis of FXR AntagonismHuang, Huang / Si, Pei / Wang, Lei / Xu, Yong / Xu, Xin / Zhu, Jin / Jiang, Hualiang / Li, Weihua / Chen, Lili / Li, Jian et al. | 2015
- 1200
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Comparative Assessment of Complex Stabilities of Radiocopper Chelating Agents by a Combination of Complex Challenge and in vivo ExperimentsLitau, Shanna / Seibold, Uwe / Vall‐Sagarra, Alicia / Fricker, Gert / Wängler, Björn / Wängler, Carmen et al. | 2015
- 1209
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Target Fishing by Cross‐Docking to Explain Polypharmacological EffectsPatel, Hitesh / Lucas, Xavier / Bendik, Igor / Günther, Stefan / Merfort, Irmgard et al. | 2015
- 1218
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Novel Furin Inhibitors with Potent Anti‐infectious ActivityHardes, Kornelia / Becker, Gero L. / Lu, Yinghui / Dahms, Sven O. / Köhler, Susanne / Beyer, Wolfgang / Sandvig, Kirsten / Yamamoto, Hiroyuki / Lindberg, Iris / Walz, Lisa et al. | 2015
- 1232
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Selective Targeting of the TPX2 Site of Importin-[alpha] Using Fragment-Based Ligand DesignRhian S Holvey et al. | 2015
- 1232
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Selective Targeting of the TPX2 Site of Importin‐α Using Fragment‐Based Ligand DesignHolvey, Rhian S. / Valkov, Eugene / Neal, David / Stewart, Murray / Abell, Chris et al. | 2015
- 1240
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Biocatalysis at Work: Applications in the Development of SagopiloneGottfried, Kathrin / Klar, Ulrich / Platzek, Johannes / Zorn, Ludwig et al. | 2015
- 1249
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Evaluation of (4‐Arylpiperidin‐1‐yl)cyclopentanecarboxamides As High‐Affinity and Long‐Residence‐Time Antagonists for the CCR2 ReceptorVilums, Maris / Zweemer, Annelien J. M. / Dilanchian, Arian / van Veldhoven, Jacobus P. D. / de Vries, Henk / Brussee, Johannes / Saunders, John / Stamos, Dean / Heitman, Laura H. / IJzerman, Adriaan P. et al. | 2015
- 1259
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Tricycloundecane Derivatives as Potential N‐Methyl‐D‐aspartate (NMDA) Receptor and Voltage‐Gated Calcium Channel ModulatorsEgunlusi, Ayodeji O. / Malan, Sarel F. / Joubert, Jacques et al. | 2015
- 1267
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Frontiers in Medicinal Chemistry 2015: Meet the Experts of MedChem near the Cradle of Medicinal and Pharmaceutical ChemistryWegscheid‐Gerlach, Christof / Gerber, Hans‐Dieter / Diederich, Wibke E. et al. | 2015
- 1273
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Human‐Based Systems for Translational Research. Edited by Robert ColemanWard, Simon E. et al. | 2015
- 1274
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Antifungals: From Genomics to Resistance and the Development of Novel Agents. Edited by Alix T. Coste and Patrick VandeputteRex, John H. et al. | 2015
- 1276
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Back Cover: Metabolic Instability of Cyanothiazolidine-Based Prolyl Oligopeptidase Inhibitors: a Structural Assignment Challenge and Potential Medicinal Chemistry ImplicationsPaolo Schiavini et al. | 2015
- 1276
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Back Cover: Metabolic Instability of Cyanothiazolidine‐Based Prolyl Oligopeptidase Inhibitors: a Structural Assignment Challenge and Potential Medicinal Chemistry Implications (ChemMedChem 7/2015)Schiavini, Paolo / Pottel, Joshua / Moitessier, Nicolas / Auclair, Karine et al. | 2015