Carbazole-containing sulfonamides and sulfamides: Discovery of cryptochrome modulators as antidiabetic agents (English)
- New search for: Steinfeld, Tod
- New search for: Steinfeld, Tod
- New search for: Kincaid, John
- New search for: Riegler, Erin
- New search for: Humphries, Paul S
- New search for: McCluskie, Kerryn
- New search for: Bersot, Ross
- New search for: Willis, Erik
- New search for: Mabery, Eric
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In:
Bioorganic & medicinal chemistry letters
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26
, 3
; 757-760
;
2016
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ISSN:
- Article (Journal) / Print
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Title:Carbazole-containing sulfonamides and sulfamides: Discovery of cryptochrome modulators as antidiabetic agents
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Contributors:Steinfeld, Tod ( author ) / Kincaid, John / Riegler, Erin / Humphries, Paul S / McCluskie, Kerryn / Bersot, Ross / Willis, Erik / Mabery, Eric / Park, Timothy / Wei, Zhi-Liang
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Published in:Bioorganic & medicinal chemistry letters ; 26, 3 ; 757-760
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Publisher:
- New search for: Elsevier
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Place of publication:Amsterdam [u.a.]
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Publication date:2016
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ISSN:
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ZDBID:
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DOI:
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Type of media:Article (Journal)
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Type of material:Print
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Language:English
- New search for: 35.70 / 44.33 / 44.42
- Further information on Basic classification
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Keywords:
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Source:
Table of contents – Volume 26, Issue 3
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 707
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Peptide-based inhibitors of protein–protein interactionsWójcik, Paulina / Berlicki, Łukasz et al. | 2015
- 714
-
Mitochondrial drug targets in neurodegenerative diseasesLee, Jiyoun et al. | 2015
- 721
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Design and discovery of new pyrimidine coupled nitrogen aromatic rings as chelating groups of JMJD3 inhibitorsHu, Jianping / Wang, Xin / Chen, Lin / Huang, Min / Tang, Wei / Zuo, Jianping / Liu, Yu-Chih / Shi, Zhe / Liu, Rongfeng / Shen, Jingkang et al. | 2016
- 726
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Growth inhibitory effect of d-arabinose against the nematode Caenorhabditis elegans: Discovery of a novel bioactive monosaccharideSakoguchi, Hirofumi / Yoshihara, Akihide / Shintani, Tomoya / Okuma, Kazuhiro / Izumori, Ken / Sato, Masashi et al. | 2016
- 730
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Bioactive lignan derivatives from the stems of Firmiana simplexWoo, Kyeong Wan / Suh, Won Se / Subedi, Lalita / Kim, Sun Yeou / Kim, Aejung / Lee, Kang Ro et al. | 2016
- 734
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Carbamate substituted 2-amino-4,6-diphenylpyrimidines as adenosine receptor antagonistsRobinson, Sarel J. / Petzer, Jacobus P. / Rousseau, Amanda L. / Terre’Blanche, Gisella / Petzer, Anél / Lourens, Anna C.U. et al. | 2016
- 739
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Toxocara canis: Larvicidal activity of fatty acid amidesMata-Santos, Taís / D’Oca, Caroline da Ros Montes / Mata-Santos, Hílton Antônio / Fenalti, Juliana / Pinto, Nitza / Coelho, Tatiane / Berne, Maria Elisabeth / da Silva, Pedro Eduardo Almeida / D’Oca, Marcelo Gonçalves Montes / Scaini, Carlos James et al. | 2016
- 742
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Discovery of imidazo[1,2-a]-pyridine inhibitors of pan-PI3 kinases that are efficacious in a mouse xenograft modelHan, Wooseok / Menezes, Daniel L. / Xu, Yongjin / Knapp, Mark S. / Elling, Robert / Burger, Matthew T. / Ni, Zhi-Jie / Smith, Aaron / Lan, Jiong / Williams, Teresa E. et al. | 2016
- 747
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Design and discovery of Novel Thiazole acetamide derivatives as anticholinesterase agent for possible role in the management of Alzheimer’sSun, Zhi-Qing / Tu, Li-Xiang / Zhuo, Feng-Juan / Liu, Song-Xia et al. | 2016
- 751
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Lead optimization of the VU0486321 series of mGlu1 PAMs. Part 2: SAR of alternative 3-methyl heterocycles and progress towards an in vivo toolGarcia-Barrantes, Pedro M. / Cho, Hyekyung P. / Metts, Adam M. / Blobaum, Anna L. / Niswender, Colleen M. / Conn, P. Jeffrey / Lindsley, Craig W. et al. | 2015
- 757
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Carbazole-containing sulfonamides and sulfamides: Discovery of cryptochrome modulators as antidiabetic agentsHumphries, Paul S. / Bersot, Ross / Kincaid, John / Mabery, Eric / McCluskie, Kerryn / Park, Timothy / Renner, Travis / Riegler, Erin / Steinfeld, Tod / Turtle, Eric D. et al. | 2015
- 761
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Antileukemic activity of lignans and phenylpropanoids of Cinnamomum parthenoxylonAdfa, Morina / Rahmad, Rizki / Ninomiya, Masayuki / Yudha S., Salprima / Tanaka, Kaori / Koketsu, Mamoru et al. | 2015
- 765
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Identification of benzothiophene amides as potent inhibitors of human nicotinamide phosphoribosyltransferaseChen, Wei / Dong, Guoqiang / He, Shipeng / Xu, Tianying / Wang, Xia / Liu, Na / Zhang, Wannian / Miao, Chaoyu / Sheng, Chunquan et al. | 2015
- 769
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The semi-synthesis of novel andrographolide analogues and anti-influenza virus activity evaluation of their derivativesYuan, Lei / Zhang, Chunfeng / Sun, Hongxin / Liu, Qingyin / Huang, Jian / Sheng, Lei / Lin, Bin / Wang, Jinhui / Chen, Lixia et al. | 2015
- 774
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Amphiphilic nanoparticles of resveratrol–norcantharidin to enhance the toxicity in zebrafish embryoYan, Deyue / Ni, Lin-Kai / Chen, Ho-Lun / Chen, Li-Chou / Chen, Yau-Hung / Cheng, Chien-Chung et al. | 2015
- 778
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Design, synthesis and in vitro activity of phidianidine B derivatives as novel PTP1B inhibitors with specific selectivityZhang, Li / Jiang, Cheng-Shi / Gao, Li-Xin / Gong, Jing-Xu / Wang, Zhong-Hua / Li, Jing-Ya / Li, Jia / Li, Xu-Wen / Guo, Yue-Wei et al. | 2015
- 782
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Structure guided design of potential inhibitors of human calcium–calmodulin dependent protein kinase IV containing pyrimidine scaffoldNaz, Huma / Jameel, Ehtesham / Hoda, Nasimul / Shandilya, Ashutosh / Khan, Parvez / Islam, Asimul / Ahmad, Faizan / Jayaram, B. / Hassan, Md. Imtaiyaz et al. | 2015
- 789
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Design, synthesis and biological evaluation of 1,3,6-trisubstituted β-carboline derivatives for cytotoxic and anti-leishmanial potentialLunagariya, Nitin A. / Gohil, Vikrantsinh M. / Kushwah, Varun / Neelagiri, Soumya / Jain, Sanyog / Singh, Sushma / Bhutani, Kamlesh K. et al. | 2015
- 795
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One-pot green synthesis of 1,3,5-triarylpentane-1,5-dione and triarylmethane derivatives as a new class of tyrosinase inhibitorsZheng, Zong-Ping / Zhang, Yi-Nan / Zhang, Shuang / Chen, Jie et al. | 2015
- 799
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Alkenes with antioxidative activities from Murraya koenigii (L.) SprengMa, Qin-Ge / Xu, Kun / Sang, Zhi-Pei / Wei, Rong-Rui / Liu, Wen-Min / Su, Ya-Lun / Yang, Jian-Bo / Wang, Ai-Guo / Ji, Teng-Fei / Li, Lu-Jun et al. | 2015
- 804
-
Synthesis and biological activity of benzamide DNA minor groove bindersKhan, Gul Shahzada / Pilkington, Lisa I. / Barker, David et al. | 2015
- 809
-
Synthesis, antimicrobial activity of Schiff base compounds of cinnamaldehyde and amino acidsWang, Hui / Yuan, Haijian / Li, Shujun / Li, Zhuo / Jiang, Mingyue et al. | 2015
- 814
-
Synthesis, anti-inflammatory, ulcerogenic and cyclooxygenase activities of indenopyrimidine derivativesUndare, Santosh S. / Valekar, Navanath J. / Patravale, Ajinkya A. / Jamale, Dattatraya K. / Vibhute, Sunil S. / Walekar, Laxman S. / Kolekar, Govind B. / Deshmukh, M.B. / Anbhule, Prashant V. et al. | 2015
- 819
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Discovery of EBI-907: A highly potent and orally active B-RafV600E inhibitor for the treatment of melanoma and associated cancersLu, Biao / Cao, Hu / Cao, Jingsong / Huang, Song / Hu, Qiyue / Liu, Dong / Shen, Ru / Shen, Xiaodong / Tao, Weikang / Wan, Hong et al. | 2015
- 824
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Identification of a small molecule HIV-1 inhibitor that targets the capsid hexamerXu, Jimmy P. / Branson, Jeffrey D. / Lawrence, Rae / Cocklin, Simon et al. | 2015
- 829
-
Antileishmanial activity of novel indolyl–coumarin hybrids: Design, synthesis, biological evaluation, molecular docking study and in silico ADME predictionSangshetti, Jaiprakash N. / Kalam Khan, Firoz A. / Kulkarni, Abhishek A. / Patil, Rajendra H. / Pachpinde, Amol M. / Lohar, Kishan S. / Shinde, Devanand B. et al. | 2015
- 836
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Synthesis, in vitro antimycobacterial evaluation and docking studies of some new 5,6,7,8-tetrahydropyrido[4′,3′:4,5]thieno[2,3-d]pyrimidin-4(3H)-one schiff basesNarender, Malothu / Jaswanth S., Bhandaru / Umasankar, Kulandaivelu / Malathi, Jojula / Raghuram Reddy, Adidala / Umadevi, K.R. / Dusthackeer, A.V.N. / Venkat Rao, Kaki / Raghuram R., Akkinepally et al. | 2015
- 841
-
Sequence selective naked-eye detection of DNA harnessing extension of oligonucleotide-modified nucleotidesVerga, Daniela / Welter, Moritz / Marx, Andreas et al. | 2015
- 845
-
Gene silencing by 2′-O-methyldithiomethyl-modified siRNA, a prodrug-type siRNA responsive to reducing environmentOchi, Yosuke / Imai, Mieko / Nakagawa, Osamu / Hayashi, Junsuke / Wada, Shun-ichi / Urata, Hidehito et al. | 2015
- 849
-
Discovery of 2-azetidinone and 1H-pyrrole-2,5-dione derivatives containing sulfonamide group at the side chain as potential cholesterol absorption inhibitorsYuan, Xinrui / Lu, Peng / Xue, Xiaojian / Qin, Hui / Fan, Chen / Wang, Yubin / Zhang, Qi et al. | 2015
- 854
-
Natural product-based synthesis of novel anti-infective isothiocyanate- and isoselenocyanate-functionalized amphilectane diterpenesNieves, Karinel / Prudhomme, Jacques / Le Roch, Karine G. / Franzblau, Scott G. / Rodríguez, Abimael D. et al. | 2015
- 858
-
Three-component, one-pot synthesis of benzo[6,7]cyclohepta[1,2-b]pyridine derivatives under catalyst free conditions and evaluation of their anti-inflammatory activitySajja, Yasodakrishna / Vulupala, Hanmanth Reddy / Bantu, Rajashaker / Nagarapu, Lingaiah / Vasamsetti, Sathish Babu / Kotamraju, Srigiridhar / Nanubolu, Jagadeesh Babu et al. | 2015
- 864
-
3D-QSAR, molecular dynamics simulations and molecular docking studies of benzoxazepine moiety as mTOR inhibitor for the treatment of lung cancerChaube, Udit / Chhatbar, Dhara / Bhatt, Hardik et al. | 2015
- 875
-
Synthesis and evaluation of an 125I-labeled azide prosthetic group for efficient and bioorthogonal radiolabeling of cyclooctyne-group containing molecules using copper-free click reactionChoi, Mi Hee / Shim, Ha Eun / Nam, You Ree / Kim, Hye Rim / Kang, Jung Ae / Lee, Dong-Eun / Park, Sang Hyun / Choi, Dae Seong / Jang, Beom-Su / Jeon, Jongho et al. | 2015
- 879
-
Mollisolactones A and B, novel dinormonoterpenes from the soft coral Sinularia mollisCheng, Shi-Yie / Wang, Shang-Kwei / Ou, Yih-Hsin / Duh, Chang-Yih et al. | 2015
- 882
-
Synthesis and positive inotropic activity evaluation of liguzinediol metabolitesZhu, Hao-hao / Chen, Yu-qing / Cheng, Dong / Li, Wei / Wang, Tian-lin / Wen, Hong-mei / Chen, Long / Liu, Jian et al. | 2015
- 885
-
Improving selectivity of dopamine D3 receptor ligandsCapet, Marc / Calmels, Thierry / Levoin, Nicolas / Danvy, Denis / Berrebi-Bertrand, Isabelle / Stark, Holger / Schwartz, Jean-Charles / Lecomte, Jeanne-Marie et al. | 2015
- 889
-
Role of the phenolic OH moiety of GluN2B-selective NMDA antagonists with 3-benzazepine scaffoldDey, Sougata / Schepmann, Dirk / Wünsch, Bernhard et al. | 2015
- 894
-
Molecular insights to the bioactive form of BV02, a reference inhibitor of 14-3-3σ protein–protein interactionsValensin, Daniela / Cau, Ylenia / Calandro, Pierpaolo / Vignaroli, Giulia / Dello Iacono, Lucia / Chiariello, Mario / Mori, Mattia / Botta, Maurizio et al. | 2015
- 899
-
TRPA1 channels as targets for resveratrol and related stilbenoidsNalli, Marianna / Ortar, Giorgio / Moriello, Aniello Schiano / Morera, Enrico / Di Marzo, Vincenzo / De Petrocellis, Luciano et al. | 2015
- 903
-
Synthesis and biological evaluation of quinoxaline di-N-oxide derivatives with in vitro trypanocidal activityPérez-Silanes, Silvia / Torres, Enrique / Arbillaga, Leire / Varela, Javier / Cerecetto, Hugo / González, Mercedes / Azqueta, Amaya / Moreno-Viguri, Elsa et al. | 2015
- 907
-
Targeting cancer cells with oleanolic and ursolic acid derived hydroxamatesWiemann, Jana / Heller, Lucie / Csuk, René et al. | 2015
- 910
-
Amides of non-steroidal anti-inflammatory drugs with thiomorpholine can yield hypolipidemic agents with improved anti-inflammatory activityTheodosis-Nobelos, Panagiotis / Kourti, Malamati / Gavalas, Antonios / Rekka, Eleni A. et al. | 2015
- 914
-
The influence of 5-HT2A activity on a 5-HT2C specific in vivo assay used for early identification of multiple acting SERT and 5-HT2C receptor ligandsÉliás, Olivér / Nógrádi, Katalin / Domány, György / Szakács, Zoltán / Kóti, János / Szántay, Csaba Jr. / Tarcsay, Ákos / Keserű, György M. / Gere, Anikó / Kiss, Béla et al. | 2015
- 921
-
Synthesis and evaluation of atorvastatin esters as prodrugs metabolically activated by human carboxylesterasesMizoi, Kenta / Takahashi, Masato / Haba, Masami / Hosokawa, Masakiyo et al. | 2015
- 924
-
Design, radiosynthesis, and evaluation of radiotracers for positron emission tomography imaging of stearoyl-CoA desaturase-1Silvers, William C. / Cai, Hancheng / Öz, Orhan K. / Sun, Xiankai et al. | 2015
- 928
-
Enantiomeric 3-deaza-1′,6′-isoneplanocin and its 3-bromo analogue: Synthesis by the Ullmann reaction and their antiviral propertiesLiu, Chong / Chen, Qi / Schneller, Stewart W. et al. | 2015
- 931
-
Discovery of potent aryl-substituted 3-[(3-methylpyridine-2-carbonyl) amino]-2,4-dimethyl-benzoic acid EP4 antagonists with improved pharmacokinetic profileBlanco, Maria-Jesus / Vetman, Tatiana / Chandrasekhar, Srinivasan / Fisher, Matthew J. / Harvey, Anita / Chambers, Mark / Lin, Chaohua / Mudra, Daniel / Oskins, Jennifer / Wang, Xu-Shan et al. | 2015
- 936
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Discovery and preclinical evaluation of potent, orally bioavailable, metabolically stable cyclopropylindolobenzazepine acylsulfonamides as thumb site 1 inhibitors of the hepatitis c virus NS5B RNA-dependent, RNA polymeraseHewawasam, Piyasena / Tu, Yong / Gao, Min / Hanumegowda, Umesh / Knipe, Jay / Lemm, Julie A. / Parker, Dawn D. / Rigat, Karen L. / Roberts, Susan B. / Meanwell, Nicholas A. et al. | 2015
- 941
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Development of curcumin–cyclodextrin/cellulose nanocrystals complexes: New anticancer drug delivery systemsNdong Ntoutoume, Gautier M.A. / Granet, Robert / Mbakidi, Jean Pierre / Brégier, Frédérique / Léger, David Y. / Fidanzi-Dugas, Chloë / Lequart, Vincent / Joly, Nicolas / Liagre, Bertrand / Chaleix, Vincent et al. | 2015
- 946
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Synthesis, structure and in vitro cytostatic activity of ferrocene—Cinchona hybridsKocsis, László / Szabó, Ildikó / Bősze, Szilvia / Jernei, Tamás / Hudecz, Ferenc / Csámpai, Antal et al. | 2015
- 950
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Structure-based design and biological evaluation of novel 2-(indol-2-yl) thiazole derivatives as xanthine oxidase inhibitorsSong, Jeong Uk / Jang, Jae Wan / Kim, Tae Hun / Park, Heuisul / Park, Wan Su / Jung, Sang-Hun / Kim, Geun Tae et al. | 2015
- 955
-
Identification of allosteric ERK2 inhibitors through in silico biased screening and competitive binding assayKinoshita, Takayoshi / Sugiyama, Hajime / Mori, Yurika / Takahashi, Naruhide / Tomonaga, Atsushi et al. | 2015
- 959
-
Receptor binding profiles and quantitative structure–affinity relationships of some 5-substituted-N,N-diallyltryptaminesCozzi, Nicholas V. / Daley, Paul F. et al. | 2015
- 965
-
Synthesis of a norcantharidin-tethered guanosine: Protein phosphatase-1 inhibitors that change alternative splicingKwiatkowski, Stefan / Sviripa, Vitaliy M. / Zhang, Zhaiyi / Wendlandt, Alison E. / Höbartner, Claudia / Watt, David S. / Stamm, Stefan et al. | 2015
- 969
-
Efficient enzymatic synthesis of l-rhamnulose and l-fuculoseWen, Liuqing / Zang, Lanlan / Huang, Kenneth / Li, Shanshan / Wang, Runling / Wang, Peng George et al. | 2015
- 973
-
Salicylates are interference compounds in TR-FRET assaysHanley, Ronan P. / Horvath, Shanti / An, Jianghong / Hof, Fraser / Wulff, Jeremy E. et al. | 2015
- 978
-
Synthesis and antituberculosis activity of indole–pyridine derived hydrazides, hydrazide–hydrazones, and thiosemicarbazonesVelezheva, Valeriya / Brennan, Patrick / Ivanov, Pavel / Kornienko, Albert / Lyubimov, Sergey / Kazarian, Konstantin / Nikonenko, Boris / Majorov, Konstantin / Apt, Alexander et al. | 2015
- 986
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Benzylamide antagonists of protease activated receptor 2 with anti-inflammatory activityYau, Mei-Kwan / Liu, Ligong / Lim, Junxian / Lohman, Rink-Jan / Cotterell, Adam J. / Suen, Jacky Y. / Vesey, David A. / Reid, Robert C. / Fairlie, David P. et al. | 2015
- 992
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A one pot, two-step synthesis of 5-arylpyrrolo[2,3-d]pyrimidines and screening of their preliminary antibacterial propertiesSaikia, Lakhinath / Roudragouda, P. / Thakur, Ashim J. et al. | 2015
- 999
-
Synthesis and evaluation of a radioiodinated 4,6-diaryl-3-cyano-2-pyridinone derivative as a survivin targeting SPECT probe for tumor imagingFuchigami, Takeshi / Mizoguchi, Tatsuya / Ishikawa, Natsumi / Haratake, Mamoru / Yoshida, Sakura / Magata, Yasuhiro / Nakayama, Morio et al. | 2015
- 1005
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Efficiently functionalized oxacalix[4]arenes: Synthesis, characterization and exploration of their biological profile as novel HDAC inhibitorsMehta, Viren / Athar, Mohd / Jha, P.C. / Panchal, Manthan / Modi, Krunal / Jain, V.K. et al. | 2015
- 1011
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Three-dimensional QSAR analysis and design of new 1,2,4-oxadiazole antibacterialsLeemans, Erika / Mahasenan, Kiran V. / Kumarasiri, Malika / Spink, Edward / Ding, Derong / O’Daniel, Peter I. / Boudreau, Marc A. / Lastochkin, Elena / Testero, Sebastian A. / Yamaguchi, Takao et al. | 2015
- 1016
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Discovery of highly potent dual EP2 and EP3 agonists with subtype selectivityKinoshita, Akihiro / Higashino, Masato / Aratani, Yoshiyuki / Kakuuchi, Akito / Matsuya, Hidekazu / Ohmoto, Kazuyuki et al. | 2015
- 1020
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Novel carbocyclic nucleoside analogs suppress glomerular mesangial cells proliferation and matrix protein accumulation through ROS-dependent mechanism in the diabetic milieu. II. Acylhydrazone-functionalized pyrimidinesBouhadir, Kamal H. / Koubeissi, Ali / Mohsen, Fatima A. / El-Harakeh, Mira Diab / Cheaib, Rouba / Younes, Joan / Azzi, Georges / Eid, Assaad A. et al. | 2015
- 1025
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A stepwise dechlorination/cross-coupling strategy to diversify the vancomycin ‘in-chloride’Wadzinski, Tyler J. / Gea, Katherine D. / Miller, Scott J. et al. | 2015
- 1029
-
Synthesis, in vitro and computational studies of 1,4-disubstituted 1,2,3-triazoles as potential α-glucosidase inhibitorsJabeen, Farukh / Shehzadi, Syeda Aaliya / Fatmi, Muhammad Qaiser / Shaheen, Sobia / Iqbal, Lubna / Afza, Nighat / Panda, Siva S. / Ansari, Farzana Latif et al. | 2015
- 1039
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Novel hydroxyamides and amides containing d-glucopyranose or d-fructose units: Biological assays in MCF-7 and MDST8 cell linesCarreiro, Elisabete P. / Costa, Ana R. / Cordeiro, Maria M. / Martins, Rute / Pires, Tiago O. / Saraiva, Mafalda / Antunes, Célia M. / Burke, Anthony J. et al. | 2015
- 1044
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2-Amino-4-bis(aryloxybenzyl)aminobutanoic acids: A novel scaffold for inhibition of ASCT2-mediated glutamine transportSchulte, Michael L. / Khodadadi, Alexandra B. / Cuthbertson, Madison L. / Smith, Jarrod A. / Manning, H. Charles et al. | 2015
- 1048
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In vitro efficacy of 2,N-bisarylated 2-ethoxyacetamides against Plasmodium falciparumGutteridge, Clare E. / Major, Joshua W. / Nin, Daniel A. / Curtis, Sean M. / Bhattacharjee, Apurba K. / Gerena, Lucia / Nichols, Daniel A. et al. | 2015
- 1052
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Multimodal formyl peptide receptor 1 targeted inflammation imaging probe: cFLFLF-MHI-DOTALi, Jie / Zhang, Yi / Chordia, Mahendra D. / Wu, Hua / Shao, Li / Pan, Dongfeng et al. | 2015
- 1056
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Adamantyl-tethered-biphenylic compounds induce apoptosis in cancer cells by targeting Bcl homologsAnusha, Sebastian / Mohan, Chakrabhavi Dhananjaya / Ananda, Hanumappa / Baburajeev, C.P. / Rangappa, Shobith / Mathai, Jessin / Fuchs, Julian E. / Li, Feng / Shanmugam, Muthu K. / Bender, Andreas et al. | 2015
- 1061
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Identification of six new lupane-type triterpenoids from Acanthopanax koreanum leaves and their tyrosinase inhibitory activitiesDat, Le Duc / Thao, Nguyen Phuong / Luyen, Bui Thi Thuy / Tai, Bui Huu / Jeong, Min Hee / Woo, Mi Hee / Kim, Young Ho et al. | 2015
- 1068
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Design, synthesis and biological evaluation of 3-substituted indenoisoquinoline derivatives as topoisomerase I inhibitorsZhao, Qian / Xu, Xi / Xie, Zhouling / Liu, Xiao / You, Qidong / Guo, Qinglong / Zhong, Yi / Li, Zhiyu et al. | 2015
- 1073
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In vitro synergistic anticancer activity of the combination of T-type calcium channel blocker and chemotherapeutic agent in A549 cellsByun, Joon Seok / Sohn, Joo Mi / Leem, Dong Gyu / Park, Byeongyeon / Nam, Ji Hye / Shin, Dong Hyun / Shin, Ji Sun / Kim, Hyoung Ja / Lee, Kyung-Tae / Lee, Jae Yeol et al. | 2015
- 1080
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Novel PTP1B inhibitors identified by DNA display of fragment pairsBarluenga, Sofia / Zambaldo, Claudio / Ioannidou, Heraklidia A. / Ciobanu, Mihai / Morieux, Pierre / Daguer, Jean-Pierre / Winssinger, Nicolas et al. | 2015
- 1086
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Fragment-based drug discovery of potent and selective MKK3/6 inhibitorsAdams, Mark / Kobayashi, Toshitake / Lawson, J. David / Saitoh, Morihisa / Shimokawa, Kenichiro / Bigi, Simone V. / Hixon, Mark S. / Smith, Christopher R. / Tatamiya, Takayuki / Goto, Masayuki et al. | 2015
- 1090
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Design and synthesis of novel selective anaplastic lymphoma kinase inhibitorsMichellys, Pierre-Yves / Chen, Bei / Jiang, Tao / Jin, Yunho / Lu, Wenshuo / Marsilje, Thomas H. / Pei, Wei / Uno, Tetsuo / Zhu, Xuefeng / Wu, Baogen et al. | 2015
- 1097
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Gambogic acid induces apoptotic cell death in T98G glioma cellsThida, Mya / Kim, Dae Won / Tran, Thi Thu Thuy / Pham, Minh Quan / Lee, Heesu / Kim, Inki / Lee, Jae Wook et al. | 2015
- IFC
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Editorial board| 2016