Cyclic RGD peptidomimetics containing 4- and 5-amino-cyclopropane pipecolic acid (CPA) templates as dual αVβ3 and α5β1 integrin ligands (English)
- New search for: Sernissi, Lorenzo
- New search for: Sernissi, Lorenzo
- New search for: Trabocchi, Andrea
- New search for: Scarpi, Dina
- New search for: Bianchini, Francesca
- New search for: Occhiato, Ernesto G
In:
Bioorganic & medicinal chemistry
;
24
, 4
; 703-711
;
2016
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ISSN:
- Article (Journal) / Print
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Title:Cyclic RGD peptidomimetics containing 4- and 5-amino-cyclopropane pipecolic acid (CPA) templates as dual αVβ3 and α5β1 integrin ligands
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Contributors:Sernissi, Lorenzo ( author ) / Trabocchi, Andrea / Scarpi, Dina / Bianchini, Francesca / Occhiato, Ernesto G
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Published in:Bioorganic & medicinal chemistry ; 24, 4 ; 703-711
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Publisher:
- New search for: Elsevier
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Place of publication:Amsterdam [u.a.]
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Publication date:2016
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ISSN:
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ZDBID:
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DOI:
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Type of media:Article (Journal)
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Type of material:Print
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Language:English
- New search for: 35.70 / 44.33 / 44.40
- Further information on Basic classification
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Source:
Table of contents – Volume 24, Issue 4
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 501
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An appraisal on recent medicinal perspective of curcumin degradant: Dehydrozingerone (DZG)Hampannavar, Girish A. / Karpoormath, Rajshekhar / Palkar, Mahesh B. / Shaikh, Mahamadhanif S. et al. | 2015
- 521
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Discovery of 2-(1H-indol-5-ylamino)-6-(2,4-difluorophenylsulfonyl)-8-methylpyrido[2,3-d]pyrimidin-7(8H)-one (7ao) as a potent selective inhibitor of Polo like kinase 2 (PLK2)Reddy, M.V. Ramana / Akula, Balireddy / Jatiani, Shashidhar / Vasquez-Del Carpio, Rodrigo / Billa, Vinay K. / Mallireddigari, Muralidhar R. / Cosenza, Stephen C. / Venkata Subbaiah, D.R.C. / Bharathi, E. Vijaya / Pallela, Venkat R. et al. | 2015
- 545
-
Active site-directed plasmin inhibitors: Extension on the P2 residueHidaka, Koushi / Gohda, Keigo / Teno, Naoki / Wanaka, Keiko / Tsuda, Yuko et al. | 2015
- 554
-
Design and synthesis of calindol derivatives as potent and selective calcium sensing receptor agonistsKiefer, Lionel / Beaumard, Floriane / Gorojankina, Tatiana / Faure, Hélène / Ruat, Martial / Dodd, Robert H. et al. | 2015
- 570
-
Allosteric inhibitors of Coxsackie virus A24 RNA polymeraseSchein, Catherine H. / Rowold, Diane / Choi, Kyung H. et al. | 2015
- 578
-
Hydroxylated chalcones with dual properties: Xanthine oxidase inhibitors and radical scavengersHofmann, Emily / Webster, Jonathan / Do, Thuy / Kline, Reid / Snider, Lindsey / Hauser, Quintin / Higginbottom, Grace / Campbell, Austin / Ma, Lili / Paula, Stefan et al. | 2015
- 588
-
Phytochemical meanings of tetrahydro-β-carboline moiety in strictosidine derivativesSudžuković, Nicole / Schinnerl, Johann / Brecker, Lothar et al. | 2015
- 596
-
Identification of B. anthracis N5-carboxyaminoimidazole ribonucleotide mutase (PurE) active site binding compounds via fragment library screeningLei, Hao / Jones, Christopher / Zhu, Tian / Patel, Kavankumar / Wolf, Nina M. / Fung, Leslie W.-M. / Lee, Hyun / Johnson, Michael E. et al. | 2015
- 606
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New hybrid molecules with anticonvulsant and antinociceptive activity derived from 3-methyl- or 3,3-dimethyl-1-[1-oxo-1-(4-phenylpiperazin-1-yl)propan-2-yl]pyrrolidine-2,5-dionesKamiński, Krzysztof / Zagaja, Mirosław / Rapacz, Anna / Łuszczki, Jarogniew J. / Andres-Mach, Marta / Abram, Michał / Obniska, Jolanta et al. | 2015
- 619
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Synthesis and biological evaluation of disubstituted amidoxanthones as potential telomeric G-quadruplex DNA-binding and apoptosis-inducing agentsShen, Rui / Chen, Yujiao / Li, Ziqian / Qi, Hui / Wang, Yitian et al. | 2015
- 627
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N-(3,4-Dimethylisoxazol-5-yl)piperazine-4-[4-(2-fluoro-4-[11C]methylphenyl)thiazol-2-yl]-1-carboxamide: A promising positron emission tomography ligand for fatty acid amide hydrolaseShimoda, Yoko / Fujinaga, Masayuki / Hatori, Akiko / Yui, Joji / Zhang, Yiding / Nengaki, Nobuki / Kurihara, Yusuke / Yamasaki, Tomoteru / Xie, Lin / Kumata, Katsushi et al. | 2015
- 635
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Synthesis, structure, and evaluation of a β-cyclodextrin-artificial carbohydrate conjugate for use as a doxorubicin-carrying moleculeYamanoi, Takashi / Oda, Yoshiki / Katsuraya, Kaname / Inazu, Toshiyuki / Hattori, Kenjiro et al. | 2015
- 643
-
Synthesis, characterization and antimicrobial activities of novel silver(I) complexes with coumarin substituted N-heterocyclic carbene ligandsKarataş, Mert Olgun / Olgundeniz, Begüm / Günal, Selami / Özdemir, İlknur / Alıcı, Bülent / Çetinkaya, Engin et al. | 2015
- 651
-
Synthesis and biological activity of ferrocenyl indeno[1,2-c]isoquinolines as topoisomerase II inhibitorsWambang, Nathalie / Schifano-Faux, Nadège / Aillerie, Alexandre / Baldeyrou, Brigitte / Jacquet, Camille / Bal-Mahieu, Christine / Bousquet, Till / Pellegrini, Sylvain / Ndifon, Peter T. / Meignan, Samuel et al. | 2015
- 661
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Illuminating the binding interactions of galactonoamidines during the inhibition of β-galactosidase (E. coli)Fan, Qiu-Hua / Pickens, Jessica B. / Striegler, Susanne / Gervaise, Cédric D. et al. | 2015
- 672
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Design, synthesis and evaluation of novel 7-aminoalkyl-substituted flavonoid derivatives with improved cholinesterase inhibitory activitiesLuo, Wen / Chen, Ying / Wang, Ting / Hong, Chen / Chang, Li-Ping / Chang, Cong-Cong / Yang, Ya-Cheng / Xie, Song-Qiang / Wang, Chao-Jie et al. | 2015
- 681
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A new chromanone derivative isolated from Hypericum lissophloeus (Hypericaceae) potentiates GABAA receptor currents in a subunit specific fashionCrockett, Sara / Baur, Roland / Kunert, Olaf / Belaj, Ferdinand / Sigel, Erwin et al. | 2015
- 686
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Design and synthesis of an activity-based protein profiling probe derived from cinnamic hydroxamic acidAi, Teng / Qiu, Li / Xie, Jiashu / Geraghty, Robert J. / Chen, Liqiang et al. | 2015
- 693
-
Synthesis and anti-tuberculosis activity of glycitylaminesCorkran, Hilary M. / Dangerfield, Emma M. / Haslett, Gregory W. / Stocker, Bridget L. / Timmer, Mattie S.M. et al. | 2015
- 703
-
Cyclic RGD peptidomimetics containing 4- and 5-amino-cyclopropane pipecolic acid (CPA) templates as dual αVβ3 and α5β1 integrin ligandsSernissi, Lorenzo / Trabocchi, Andrea / Scarpi, Dina / Bianchini, Francesca / Occhiato, Ernesto G. et al. | 2015
- 712
-
Synthesis and biological evaluation of novel 5-hydroxylaminoisoxazole derivatives as lipoxygenase inhibitors and metabolism enhancing agentsAverina, Elena B. / Vasilenko, Dmitry A. / Gracheva, Yulia A. / Grishin, Yuri K. / Radchenko, Eugene V. / Burmistrov, Vladimir V. / Butov, Gennady M. / Neganova, Margarita E. / Serkova, Tatyana P. / Redkozubova, Olga M. et al. | 2015
- 721
-
New MKLP-2 inhibitors in the paprotrain series: Design, synthesis and biological evaluationsLabrière, Christophe / Talapatra, Sandeep K. / Thoret, Sylviane / Bougeret, Cécile / Kozielski, Frank / Guillou, Catherine et al. | 2015
- 735
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Synthesis of novel polybrominated benzimidazole derivatives—potential CK2 inhibitors with anticancer and proapoptotic activityŁukowska-Chojnacka, Edyta / Wińska, Patrycja / Wielechowska, Monika / Poprzeczko, Martyna / Bretner, Maria et al. | 2015
- 742
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Three new double-headed nucleotides with additional nucleobases connected to C-5 of pyrimidines; synthesis, duplex and triplex studiesKumar, Pawan / Sharma, Pawan K. / Hansen, Jonas / Jedinak, Lukas / Reslow-Jacobsen, Charlotte / Hornum, Mick / Nielsen, Poul et al. | 2015
- 750
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Expanding the structural diversity of diarylureas as multi-target tyrosine kinase inhibitorsShan, Yuanyuan / Wang, Chen / Zhang, Lin / Wang, Jinfeng / Wang, Maoyi / Dong, Yalin et al. | 2015
- 759
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Structural features underlying raloxifene’s biophysical interaction with bone matrixBivi, Nicoletta / Hu, Haitao / Chavali, Balagopalakrishna / Chalmers, Michael J. / Reutter, Christopher T. / Durst, Gregory L. / Riley, Anna / Sato, Masahiko / Allen, Matthew R. / Burr, David B. et al. | 2015
- 768
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Investigating molecular dynamics-guided lead optimization of EGFR inhibitorsLavecchia, Martin J. / Puig de la Bellacasa, Raimon / Borrell, José I. / Cavasotto, Claudio N. et al. | 2015
- 779
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Synthesis and biological evaluation of 3-tetrazolo steroidal analogs: Novel class of 5α-reductase inhibitorsAggarwal, Saurabh / Mahapatra, Manoj Kumar / Kumar, Rajnish / Bhardwaj, Tilak R. / Hartmann, Rolf W. / Haupenthal, Jörg / Kumar, Manoj et al. | 2015
- 789
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Design and synthesis of novel androgen receptor antagonists via molecular modelingZhao, Chao / Choi, You Hee / Khadka, Daulat Bikram / Jin, Yifeng / Lee, Kwang-Youl / Cho, Won-Jea et al. | 2015
- 802
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Synthesis, isomerization and biological activity of novel 2-selenohydantoin derivativesIvanenkov, Yan A. / Veselov, Mark S. / Rezekin, Igor G. / Skvortsov, Dmitriy A. / Sandulenko, Yuri B. / Polyakova, Marina V. / Bezrukov, Dmitry S. / Vasilevsky, Sergey V. / Kukushkin, Maxim E. / Moiseeva, Anna A. et al. | 2015
- 812
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Design, synthesis, and docking studies of phenylpicolinamide derivatives bearing 1H-pyrrolo[2,3-b]pyridine moiety as c-Met inhibitorsZhu, Wufu / Wang, Wenhui / Xu, Shan / Tang, Qidong / Luo, Rong / Wang, Min / Gong, Ping / Zheng, Pengwu et al. | 2016
- 820
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2,3-Dihydrobenzofuran privileged structures as new bioinspired lead compounds for the design of mPGES-1 inhibitorsDi Micco, Simone / Spatafora, Carmela / Cardullo, Nunzio / Riccio, Raffaele / Fischer, Katrin / Pergola, Carlo / Koeberle, Andreas / Werz, Oliver / Chalal, Malik / Vervandier-Fasseur, Dominique et al. | 2016
- 827
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Synthesis and evaluation of styrylpyran fluorophores for noninvasive detection of cerebral β-amyloid depositsZhu, Bi-yue / Cheng, Yan / Li, Guo-bo / Yang, Sheng-yong / Zhang, Zhi-rong et al. | 2016
- 835
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Cloning, characterization and anion inhibition studies of a γ-carbonic anhydrase from the Antarctic bacterium Colwellia psychrerythraeaDe Luca, Viviana / Vullo, Daniela / Del Prete, Sonia / Carginale, Vincenzo / Osman, Sameh M. / AlOthman, Zeid / Supuran, Claudiu T. / Capasso, Clemente et al. | 2016
- 841
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Synthesis, antimicrobial evaluation and molecular modeling of 5-hydroxyisoquinolinium salt series; the effect of the hydroxyl moietySoukup, Ondrej / Dolezal, Rafael / Malinak, David / Marek, Jan / Salajkova, Sarka / Pasdiorova, Marketa / Honegr, Jan / Korabecny, Jan / Nachtigal, Petr / Nachon, Florian et al. | 2016
- 849
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Novel triazolothiadiazines act as potent anticancer agents in liver cancer cells through Akt and ASK-1 proteinsAytaç, Peri S. / Durmaz, Irem / Houston, Douglas R. / Çetin-Atalay, Rengül / Tozkoparan, Birsen et al. | 2016
- 873
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- 877
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- 886
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Ferulic acid–carbazole hybrid compounds: Combination of cholinesterase inhibition, antioxidant and neuroprotection as multifunctional anti-Alzheimer agentsFang, Lei / Chen, Mohao / Liu, Zhikun / Fang, Xubin / Gou, Shaohua / Chen, Li et al. | 2016
- 894
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Sulfamide derivatives with selective carbonic anhydrase VII inhibitory actionVillalba, Maria Luisa / Palestro, Pablo / Ceruso, Mariangela / Gonzalez Funes, Jose L. / Talevi, Alan / Bruno Blanch, Luis / Supuran, Claudiu T. / Gavernet, Luciana et al. | 2016
- 902
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Fluorinated matrix metalloproteinases inhibitors—Phosphonate based potential probes for positron emission tomographyBeutel, Bernd / Daniliuc, Constantin G. / Riemann, Burkhard / Schäfers, Michael / Haufe, Günter et al. | 2016
- 910
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DNA cleavage at the AP site via β-elimination mediated by the AP site-binding ligandsAbe, Yukiko S. / Sasaki, Shigeki et al. | 2016
- 915
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Synthesis and immunological evaluation of N-acyl modified Tn analogues as anticancer vaccine candidatesSong, Chengcheng / Sun, Shuang / Huo, Chang-Xin / Li, Qin / Zheng, Xiu-Jing / Tai, Guihua / Zhou, Yifa / Ye, Xin-Shan et al. | 2016
- 921
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- IFC
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Editorial board| 2016