Novel naphtho[2,1-d]oxazole-4,5-diones as NQO1 substrates with improved aqueous solubility: Design, synthesis, and in vivo antitumor evaluation (English)
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In:
Bioorganic & medicinal chemistry
;
24
, 5
; 1006-1013
;
2016
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ISSN:
- Article (Journal) / Print
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Title:Novel naphtho[2,1-d]oxazole-4,5-diones as NQO1 substrates with improved aqueous solubility: Design, synthesis, and in vivo antitumor evaluation
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Contributors:Li, Xiang ( author ) / Bian, Jinlei / Wang, Nan / Qian, Xue / Gu, Jing / Mu, Tong / Fan, Jun / Yang, Xiuwen / Li, Shangzhen / Yang, Tingting
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Published in:Bioorganic & medicinal chemistry ; 24, 5 ; 1006-1013
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Publisher:
- New search for: Elsevier
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Place of publication:Amsterdam [u.a.]
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Publication date:2016
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ISSN:
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ZDBID:
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DOI:
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Type of media:Article (Journal)
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Type of material:Print
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Language:English
- New search for: 35.70 / 44.33 / 44.40
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Source:
Table of contents – Volume 24, Issue 5
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 929
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A spectroscopic study of substituted anthranilic acids as sensitive environmental probes for detecting cancer cellsCulf, Adrian S. / Yin, Huimin / Monro, Susan / Ghosh, Anirban / Barnett, David A. / Ouellette, Rodney J. / Čuperlović-Culf, Miroslava / McFarland, Sherri A. et al. | 2015
- 938
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Design, synthesis, and biological evaluation of water-soluble amino acid prodrug conjugates derived from combretastatin, dihydronaphthalene, and benzosuberene-based parent vascular disrupting agentsDevkota, Laxman / Lin, Chen-Ming / Strecker, Tracy E. / Wang, Yifan / Tidmore, Justin K. / Chen, Zhi / Guddneppanavar, Rajsekhar / Jelinek, Christopher J. / Lopez, Ramona / Liu, Li et al. | 2016
- 957
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Discovery of benzenesulfonamide derivatives as potent PI3K/mTOR dual inhibitors with in vivo efficacies against hepatocellular carcinomaChen, Ying / Zhang, Ling / Yang, Chao / Han, Jinsong / Wang, Chongqing / Zheng, Canhui / Zhou, Youjun / Lv, Jiaguo / Song, Yunlong / Zhu, Ju et al. | 2016
- 967
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Overcoming multidrug resistance by targeting mitochondria with NO-donating doxorubicinsGazzano, Elena / Chegaev, Konstantin / Rolando, Barbara / Blangetti, Marco / Annaratone, Lorenzo / Ghigo, Dario / Fruttero, Roberta / Riganti, Chiara et al. | 2016
- 976
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Kinetic and X-ray crystallographic investigations on carbonic anhydrase isoforms I, II, IX and XII of a thioureido analog of SLC-0111Lomelino, Carrie L. / Mahon, Brian P. / McKenna, Robert / Carta, Fabrizio / Supuran, Claudiu T. et al. | 2016
- 982
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Synthesis of 4-sulfamoylphenyl-benzylamine derivatives with inhibitory activity against human carbonic anhydrase isoforms I, II, IX and XIIDurgun, Mustafa / Turkmen, Hasan / Ceruso, Mariangela / Supuran, Claudiu T. et al. | 2016
- 989
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Insight to the binding mode of triazole RGD-peptidomimetics to integrin-rich cancer cells by NMR and molecular modelingVasile, Francesca / Menchi, Gloria / Lenci, Elena / Guarna, Antonio / Potenza, Donatella / Trabocchi, Andrea et al. | 2016
- 995
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Anionic surfactants enhance click reaction-mediated protein conjugation with ubiquitinSchneider, Daniel / Schneider, Tatjana / Aschenbrenner, Joos / Mortensen, Franziska / Scheffner, Martin / Marx, Andreas et al. | 2016
- 1002
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In vitro interactions between anidulafungin and nonsteroidal anti-inflammatory drugs on biofilms of Candida spp.Rosato, Antonio / Catalano, Alessia / Carocci, Alessia / Carrieri, Antonio / Carone, Addolorata / Caggiano, Giuseppina / Franchini, Carlo / Corbo, Filomena / Montagna, Maria Teresa et al. | 2016
- 1006
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Novel naphtho[2,1-d]oxazole-4,5-diones as NQO1 substrates with improved aqueous solubility: Design, synthesis, and in vivo antitumor evaluationLi, Xiang / Bian, Jinlei / Wang, Nan / Qian, Xue / Gu, Jing / Mu, Tong / Fan, Jun / Yang, Xiuwen / Li, Shangzhen / Yang, Tingting et al. | 2016
- 1014
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Discovery of novel phenoxazinone derivatives as DKK1/LRP6 interaction inhibitors: Synthesis, biological evaluation and structure–activity relationshipsThysiadis, Savvas / Mpousis, Spyros / Avramidis, Nicolaos / Katsamakas, Sotirios / Balomenos, Athanasios / Remelli, Rosaria / Efthimiopoulos, Spyros / Sarli, Vasiliki et al. | 2016
- 1023
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Discovery of potent anti-tuberculosis agents targeting leucyl-tRNA synthetaseGudzera, Olga I. / Golub, Andriy G. / Bdzhola, Volodymyr G. / Volynets, Galyna P. / Lukashov, Sergiy S. / Kovalenko, Oksana P. / Kriklivyi, Ivan A. / Yaremchuk, Anna D. / Starosyla, Sergiy A. / Yarmoluk, Sergiy M. et al. | 2016
- 1032
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Synthesis and biological evaluation of enantiomerically pure glyceric acid derivatives as LpxC inhibitorsTangherlini, Giovanni / Torregrossa, Tullio / Agoglitta, Oriana / Köhler, Jens / Melesina, Jelena / Sippl, Wolfgang / Holl, Ralph et al. | 2016
- 1045
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Incorporation of fluorophore–cholesterol conjugates into liposomal and mycobacterial membranesWercholuk, Ashley N. / Thuman, Jenna M. / Stanley, Jordan L. / Sargent, Andrew L. / Anderson, Eric S. / Allen, William E. et al. | 2016
- 1050
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Synthesis, molecular docking and biological evaluation of N,N-disubstituted 2-aminothiazolines as a new class of butyrylcholinesterase and carboxylesterase inhibitorsMakhaeva, Galina F. / Boltneva, Natalia P. / Lushchekina, Sofya V. / Serebryakova, Olga G. / Stupina, Tatyana S. / Terentiev, Alexey A. / Serkov, Igor V. / Proshin, Alexey N. / Bachurin, Sergey O. / Richardson, Rudy J. et al. | 2016
- 1063
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Pyrazole antagonists of the CB1 receptor with reduced brain penetrationFulp, Alan / Zhang, Yanan / Bortoff, Katherine / Seltzman, Herbert / Snyder, Rodney / Wiethe, Robert / Amato, George / Maitra, Rangan et al. | 2016
- 1071
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A clickable psoralen to directly quantify DNA interstrand crosslinking and repairEvison, Benjamin J. / Actis, Marcelo L. / Fujii, Naoaki et al. | 2016
- 1079
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Synthesis and pharmacological evaluation of trifluoromethyl containing 4-(2-pyrimidinylamino)benzamides as Hedgehog signaling pathway inhibitorsXin, Minhang / Zhang, Liandi / Wen, Jun / Shen, Han / Liu, Zhaoyu / Zhao, Xinge / Jin, Qiu / Wang, Mengyu / Cheng, Lingfei / Huang, Wei et al. | 2016
- 1089
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Symmetric 4,4′-(piperidin-4-ylidenemethylene)bisphenol derivatives as novel tunable estrogen receptor (ER) modulatorsSato, Manabu / Ohta, Kiminori / Kaise, Asako / Aoto, Sayaka / Endo, Yasuyuki et al. | 2016
- 1095
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A novel library of saccharin and acesulfame derivatives as potent and selective inhibitors of carbonic anhydrase IX and XII isoformsCarradori, Simone / Secci, Daniela / De Monte, Celeste / Mollica, Adriano / Ceruso, Mariangela / Akdemir, Atilla / Sobolev, Anatoly P. / Codispoti, Rossella / De Cosmi, Federica / Guglielmi, Paolo et al. | 2016
- 1106
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Heptapeptide ligands against receptor-binding sites of influenza hemagglutinin toward anti-influenza therapyMatsubara, Teruhiko / Onishi, Ai / Yamaguchi, Daisuke / Sato, Toshinori et al. | 2016
- 1115
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Sulfonamide inhibition studies of the β-carbonic anhydrase from the pathogenic bacterium Vibrio choleraeDel Prete, Sonia / Vullo, Daniela / De Luca, Viviana / Carginale, Vincenzo / Ferraroni, Marta / Osman, Sameh M. / AlOthman, Zeid / Supuran, Claudiu T. / Capasso, Clemente et al. | 2016
- 1121
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Metal-based biologically active azoles and β-lactams derived from sulfa drugsEbrahimi, Hossein Pasha / Hadi, Jabbar S. / Almayah, Abdulelah A. / Bolandnazar, Zeinab / Swadi, Ali G. / Ebrahimi, Amirpasha et al. | 2016
- 1132
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Glycopeptide-functionalized gold nanoparticles for antibody induction against the tumor associated mucin-1 glycoproteinCai, Hui / Degliangeli, Federica / Palitzsch, Björn / Gerlitzki, Bastian / Kunz, Horst / Schmitt, Edgar / Fiammengo, Roberto / Westerlind, Ulrika et al. | 2016
- 1136
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Structure–activity relationship study of 4-(thiazol-5-yl)benzoic acid derivatives as potent protein kinase CK2 inhibitorsOhno, Hiroaki / Minamiguchi, Daiki / Nakamura, Shinya / Shu, Keito / Okazaki, Shiho / Honda, Maho / Misu, Ryosuke / Moriwaki, Hirotomo / Nakanishi, Shinsuke / Oishi, Shinya et al. | 2016
- 1142
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Synthesis and cytotoxicity of thieno[2,3-b]quinoline-2-carboxamide and cycloalkyl[b]thieno[3,2-e]pyridine-2-carboxamide derivativesLeung, Euphemia / Pilkington, Lisa I. / van Rensburg, Michelle / Jeon, Chae Yeon / Song, Mirae / Arabshahi, Homayon J. / De Zoysa, Gayan Heruka / Sarojini, Vijayalekshmi / Denny, William A. / Reynisson, Jóhannes et al. | 2016
- 1155
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Assemblies of ionic zinc chlorins assisted by water-soluble polypeptidesMiyatake, Tomohiro / Hasunuma, Yuki / Mukai, Yumi / Oki, Hisato / Watanabe, Mikiya / Yamazaki, Shohei et al. | 2016
- IFC
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Editorial board| 2016