Optimization and multigram scalability of a catalytic enantioselective borylative migration for the synthesis of functionalized chiral piperidinesElectronic supplementary information (ESI) available: 1H and 13C NMR spectra of new compounds and experimental procedures. See DOI: 10.1039/c6ob00685j (English)
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Organic & biomolecular chemistry
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14
, 2
; 4739-4748
;
2016
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ISSN:
- Article (Journal) / Print
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Title:Optimization and multigram scalability of a catalytic enantioselective borylative migration for the synthesis of functionalized chiral piperidinesElectronic supplementary information (ESI) available: 1H and 13C NMR spectra of new compounds and experimental procedures. See DOI: 10.1039/c6ob00685j
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Contributors:Kim, You-Ri ( author ) / Hall, Dennis G
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Published in:Organic & biomolecular chemistry ; 14, 2 ; 4739-4748
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- New search for: RSC
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Place of publication:Cambridge
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Publication date:2016
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Type of media:Article (Journal)
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Type of material:Print
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Language:English
- New search for: 35.70 / 35.70 / 35.50 / 35.50
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Source:
Table of contents – Volume 14, Issue 2
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 43
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A protocol for amide bond formation with electron deficient amines and sterically hindered substratesElectronic supplementary information (ESI) available: Synthetic procedures, compound characterization, NMR spectra. See DOI: 10.1039/c5ob02129dDue-Hansen, Maria E et al. | 2015
- 44
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Targeting anti-apoptotic Bcl2 proteins with scyllatoxin-based BH3 domain mimeticsElectronic supplementary information (ESI) available: Supporting figures and experimental details. See DOI: 10.1039/c5ob02080hHarris, M. Margaret et al. | 2015
- 46
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Formal synthesis of (−)-podophyllotoxin through the photocyclization of an axially chiral 3,4-bisbenzylidene succinate amide ester - a flow photochemistry approachElectronic supplementary information (ESI) available: NMR, UV spectra, photo of the system for "in-flow" photoreactions and crystallographic data. CCDC 1415848. For ESI and crystallographic data in CIF or other electronic format see DOI: 10.1039/c5ob01844gLisiecki, Kamil et al. | 2015
- 47
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[1,4]-sigmatropic rearrangement of chiral nitrones and their utilization in the synthesis of new iminosugarsElectronic supplementary information (ESI) available: Copies of 1H and 13C NMR spectra of all new compounds, details of biological activity tests, X-ray structure determination details and crystallographic data (CIF files) for alcohol 13 and indolizidine 15a hydrochloride, absolute (Hartrees) and relative (kcal mol−1) electronic and free energies and Cartesian coordinates of all optimized structures. CCDC 1410262 and 1410265. For ESI and crystallographic data in CIF or other electronic format see DOI: 10.1039/c5ob01432hMalinowski, Maciej et al. | 2015
- 409
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Alkaloid synthesis using chiral secondary amine organocatalystsIshikawa, Hayato / Shiomi, Shinya et al. | 2015
- 53
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Synthesis of a new β-amino acid with a 3-deoxy-l-ara furnaoside side chain: the influence of the side chain on the conformation of α/β-peptidesElectronic supplementary information (ESI) available. See DOI: 10.1039/c5ob01753jSharma, Gangavaram V. M et al. | 2015
- 57
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A concentration dependent auto-relay-recognition by the same analyte: a dual fluorescence switch-on by hydrogen sulfide via Michael addition followed by reduction and staining for bio-activityElectronic supplementary information (ESI) available: Detailed synthesis procedure of the probes, NMR, HRMS, experimental details, computational data etc. See DOI: 10.1039/c5ob02008eDas, Avijit Kumar et al. | 2015
- 59
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Iodine-catalyzed expeditious synthesis of sulfonamides from sulfonyl hydrazides and aminesElectronic supplementary information (ESI) available. See DOI: 10.1039/c5ob02075aYotphan, Sirilata et al. | 2015
- 68
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Design, synthesis and evaluation of N-aryl-glyoxamide derivatives as structurally novel bacterial quorum sensing inhibitorsElectronic supplementary information (ESI) available: NMR spectra of synthesized compounds and bacterial growth inhibition data. See DOI: 10.1039/c5ob01973gNizalapur, Shashidhar et al. | 2015
- 71
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Molecular construction of HIV-gp120 discontinuous epitope mimics by assembly of cyclic peptides on an orthogonal alkyne functionalized TAC-scaffoldElectronic supplementary information (ESI) available: Analytical data for peptides, constructs and intermediates. See DOI: 10.1039/c5ob02014jWerkhoven, P. R et al. | 2015
- 373
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Front cover| 2015
- 374
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Inside front cover| 2015
- 375
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Contents list| 2015
- 389
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Fluorinated porphyrinoids as efficient platforms for new photonic materials, sensors, and therapeuticsBhupathiraju, N. V. S. Dinesh K. / Rizvi, Waqar / Batteas, James D. / Drain, Charles Michael et al. | 2015
- 425
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On the association of neutral and cationic tris(tetrathiafulvaleno)dodecadehydro[18]annulenesParker, Christian R. / Lincke, Kasper / Christensen, Mikkel A. / Lušpai, Karol / Rapta, Peter / Sørensen, Thomas Just / Morsing, Thorbjørn J. / Du, Lin / Kjaergaard, Henrik G. / Hammerich, Ole et al. | 2015
- 430
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A protocol for amide bond formation with electron deficient amines and sterically hindered substratesDue-Hansen, Maria E. / Pandey, Sunil K. / Christiansen, Elisabeth / Andersen, Rikke / Hansen, Steffen V. F. / Ulven, Trond et al. | 2015
- 434
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Metal-free Brønsted acid mediated synthesis of fully substituted thiophenes via chemo- and regioselective intramolecular cyclization of α,α′-bis(β-oxodithioesters) at room temperatureRamulu, B. Janaki / Koley, Suvajit / Singh, Maya Shankar et al. | 2015
- 434
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Metal-free Bronsted acid mediated synthesis of fully substituted thiophenes via chemo- and regioselective intramolecular cyclization of a,aprime-bis(b-oxodithioesters) at room temperatureRamulu, B. J. / Koley, S. / Singh, M. et al. | 2016
- 440
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Targeting anti-apoptotic Bcl2 proteins with scyllatoxin-based BH3 domain mimeticsHarris, M. Margaret / Coon, Zachary / Alqaeisoom, Najah / Swords, Brian / Holub, Justin M. et al. | 2015
- 447
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The dual aptamer approach: rational design of a high-affinity FAD aptamerMerkle, T. / Holder, I. T. / Hartig, J. S. et al. | 2015
- 451
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Pd-indenyl-diphosphine: an effective catalyst for the preparation of triarylaminesYan, Meng-Qi / Yuan, Jia / Pi, Yun-Xiao / Liang, Jin-Hua / Liu, Yan / Wu, Qing-Guo / Luo, Xue / Liu, Sheng-Hua / Chen, Jian / Zhu, Xiao-Lei et al. | 2015
- 455
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Photochemically re-bridging disulfide bonds and the discovery of a thiomaleimide mediated photodecarboxylation of C-terminal cysteinesRichards, Daniel A. / Fletcher, Sally A. / Nobles, Muriel / Kossen, Hanno / Tedaldi, Lauren / Chudasama, Vijay / Tinker, Andrew / Baker, James R. et al. | 2015
- 459
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Zwitterionic [4]helicene: a water-soluble and reversible pH-triggered ECD/CPL chiroptical switch in the UV and red spectral regionsElectronic supplementary information (ESI) available: Solubility study, pKa determination, characterization of M/P enantiomers, additional optical, chiroptical and theoretical data. CCDC 1472769. For ESI and crystallographic data in CIF or other electronic format see DOI: 10.1039/c6ob00752jPascal, Simon et al. | 2016
- 460
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Formal synthesis of (−)-podophyllotoxin through the photocyclization of an axially chiral 3,4-bisbenzylidene succinate amide ester – a flow photochemistry approachLisiecki, Kamil / Krawczyk, Krzysztof K. / Roszkowski, Piotr / Maurin, Jan K. / Czarnocki, Zbigniew et al. | 2015
- 464
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Nucleoside-2,3/3,5-bis(thio)phosphate antioxidants are also capable of disassembly of amyloid beta42-Zn(ii)/Cu(ii) aggregates via Zn(ii)/Cu(ii)-chelationElectronic supplementary information (ESI) available. See DOI: 10.1039/c6ob00613bHevroni, Bosmat Levi et al. | 2016
- 465
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Development of novel PP2A activators for use in the treatment of acute myeloid leukaemiaElectronic supplementary information (ESI) available: Synthetic procedures and characterisation data for all new compounds. See DOI: 10.1039/c6ob00556jToop, Hamish D et al. | 2016
- 469
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Concise total synthesis of (±)-serotobenineElectronic supplementary information (ESI) available: 1NMR and 13NMR spectra. See DOI: 10.1039/c6ob00682eLiang, Kangjiang et al. | 2016
- 470
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[1,4]-sigmatropic rearrangement of chiral nitrones and their utilization in the synthesis of new iminosugarsMalinowski, Maciej / Rowicki, Tomasz / Guzik, Patrycja / Gryszel, Maciej / Łapczyński, Sebastian / Wielechowska, Monika / Czerwińska, Karolina / Madura, Izabela / Sas, Wojciech et al. | 2015
- 474
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Brønsted base-catalyzed three-component coupling reaction of -ketoesters, imines, and diethyl phosphite utilizing [1,2]-phospha-Brook rearrangementElectronic supplementary information (ESI) available: Experimental procedures and characterization data. CCDC 1046578 and 1450154. For ESI and crystallographic data in CIF or other electronic format see DOI: 10.1039/c6ob00739bKondoh, Azusa et al. | 2016
- 483
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Synthesis and characterisation of a mesocyclic tripodal triamine ligandUre, Andrew D. / Lázaro, Isabel Abánade / Cotter, Michelle / McDonald, Aidan R. et al. | 2015
- 495
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Synthesis of 3,3prime-carbonyl-bis(chromones) and their activity as mammalian alkaline phosphatase inhibitorsMiliutina, M. / Ejaz, S. / Iaroshenko, V. / Villinger, A. / Iqbal, J. / Langer, P. et al. | 2016
- 495
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Synthesis of 3,3′-carbonyl-bis(chromones) and their activity as mammalian alkaline phosphatase inhibitorsMiliutina, Mariia / Ejaz, Syeda Abida / Iaroshenko, Viktor O. / Villinger, Alexander / Iqbal, Jamshed / Langer, Peter et al. | 2015
- 503
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Synthesis of a new b-amino acid with a 3-deoxy-L-ara furnaoside side chain: the influence of the side chain on the conformation of a/b-peptidesSharma, G. M. / Anjaiah, G. / Kanakaraju, M. / Sudhakar, B. / Chatterjee, D. / Kunwar, A. et al. | 2016
- 503
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Synthesis of a new β-amino acid with a 3-deoxy-l-ara furnaoside side chain: the influence of the side chain on the conformation of α/β-peptidesSharma, Gangavaram V. M. / Anjaiah, Gonuguntla / Kanakaraju, Marumudi / Sudhakar, Bommeda / Chatterjee, Deepak / Kunwar, Ajit C. et al. | 2015
- 516
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Selective modification of the 3′′-amino group of kanamycin prevents significant loss of activity in resistant bacterial strainsSantana, Andrés G. / Zárate, Sandra G. / Asensio, Juan Lui / Revuelta, Julia / Bastida, Agatha et al. | 2015
- 516
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Selective modification of the 3primeprime-amino group of kanamycin prevents significant loss of activity in resistant bacterial strainsSantana, A. / Zarate, S. / Asensio, J. / Revuelta, J. / Bastida, A. et al. | 2016
- 526
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Selective synthesis of functionalized pyrroles from 3-aza-1,5-enynesZhao, Yingying / Wang, Haolong / Li, Xincheng / Wang, Dongping / Xin, Xiaoyi / Wan, Boshun et al. | 2015
- 542
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DNA bases ring-expanded with a cyclopentadiene free radical: a theoretical investigation of building blocks with diradical characterZhao, Peiwen / Bu, Yuxiang et al. | 2015
- 556
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A facile one pot route for the synthesis of imide tethered peptidomimeticsPanduranga, Veladi / Prabhu, Girish / Kumar, Roopesh / Basavaprabhu, / Sureshbabu, Vommina V. et al. | 2015
- 564
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Synthesis of α-haloenamides via zinc halide mediated direct addition of benzhydryl halides to ynamidesChen, Ling / Yu, Lian / Deng, Yuan / Cui, Yuming / Bian, Gaofeng / Cao, Jian et al. | 2015
- 564
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Synthesis of a-haloenamides via zinc halide mediated direct addition of benzhydryl halides to ynamidesChen, L. / Yu, L. / Deng, Y. / Cui, Y. / Bian, G. / Cao, J. et al. | 2016
- 570
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A concentration dependent auto-relay-recognition by the same analyte: a dual fluorescence switch-on by hydrogen sulfide via Michael addition followed by reduction and staining for bio-activityDas, Avijit Kumar / Goswami, Shyamaprosad / Dutta, Gorachand / Maity, Sibaprasad / Mandal, Tarun kanti / Khanra, Kalyani / Bhattacharyya, Nandan et al. | 2015
- 577
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AIBN/NaBr-promoted aerobic oxidation of benzylic alcohols via a radical processLiu, Chengkou / Fang, Zheng / Yang, Zhao / Li, Qingwen / Guo, Shiyu / Guo, Kai et al. | 2015
- 582
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One pot oxidative N–S bond formation to access 2-sulfenylimine chromenesKale, Ashok / Chennapuram, Madhu / Bingi, Chiranjeevi / Nanubolu, Jagadeesh Babu / Atmakur, Krishnaiah et al. | 2015
- 590
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Iodine-catalyzed expeditious synthesis of sulfonamides from sulfonyl hydrazides and aminesYotphan, Sirilata / Sumunnee, Ladawan / Beukeaw, Danupat / Buathongjan, Chonchanok / Reutrakul, Vichai et al. | 2015
- 598
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The synthesis of heterosaccharides related to the fucoidan from Chordaria flagelliformis bearing an α-l-fucofuranosyl unitVinnitskiy, Dmitry Z. / Krylov, Vadim B. / Ustyuzhanina, Nadezhda E. / Dmitrenok, Andrey S. / Nifantiev, Nikolay E. et al. | 2015
- 598
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The synthesis of heterosaccharides related to the fucoidan from Chordaria flagelliformis bearing an a-L-fucofuranosyl unitVinnitskiy, D. / Krylov, V. / Ustyuzhanina, N. / Dmitrenok, A. / Nifantiev, N. et al. | 2016
- 612
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A study on the AMACR catalysed elimination reaction and its application to inhibitor testingYevglevskis, Maksim / Lee, Guat L. / Sun, Jenny / Zhou, Shiyi / Sun, Xiaolong / Kociok-Köhn, Gabriele / James, Tony D. / Woodman, Timothy J. / Lloyd, Matthew D. et al. | 2015
- 623
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Effective and novel enantioselective preparation of pyranopyrazoles and pyranocoumarins that is catalyzed by a quinine-derived primary amineYang, Sai / Shen, Liu-lan / Kim, Yoon-Jung / Jeong, Jin-Hyun et al. | 2015
- 631
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Design of a fluorescent ligand targeting the S-adenosylmethionine binding site of the histone methyltransferase MLL1Luan, Yepeng / Blazer, Levi L. / Hu, Hao / Hajian, Taraneh / Zhang, Jing / Wu, Hong / Houliston, Scott / Arrowsmith, Cheryl H. / Vedadi, Masoud / Zheng, Yujun George et al. | 2015
- 639
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An efficient synthesis of an exo-enone analogue of LL-Z1640-2 and evaluation of its protein kinase inhibitory activitiesWang, Stephanie Q. / Goh, Shermin S. / Chai, Christina L. L. / Chen, Anqi et al. | 2015
- 646
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Epigenetic stimulation of polyketide production in Chaetomium cancroideum by an NAD+-dependent HDAC inhibitorAsai, Teigo / Morita, Shuntaro / Taniguchi, Tohru / Monde, Kenji / Oshima, Yoshiteru et al. | 2015
- 652
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Effective chemiluminogenic systems based on acridinium esters bearing substituents of various electronic and steric propertiesZadykowicz, Beata / Czechowska, Justyna / Ożóg, Agnieszka / Renkevich, Anton / Krzymiński, Karol et al. | 2015
- 669
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Readily prepared inclusion forming chiral calixsalensJaniak, Agnieszka / Petryk, Małgorzata / Barbour, Leonard J. / Kwit, Marcin et al. | 2015
- 669
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Readily prepared inclusion forming chiral calixsalensElectronic supplementary information (ESI) available: Details of the synthesis of 3a-3g, along with general experimental protocols and detailed descriptions of the crystallographic procedures and structures. CCDC 1422957 (3a), 1422958 (3b), 1422959 (3c), 1422960 (3d), 1422961 (3e), 1422962 (3f), 1422963 (3fsCO2), 1422964 (3g) and 1422965 (3gMeCN). For ESI and crystallographic data in CIF or other electronic format see DOI: 10.1039/c5ob02090eJaniak, Agnieszka et al. | 2015
- 674
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Host–guest complexation of di-cyclohexanocucurbit[6]uril and hexa-cyclohexanocucurbit[6]uril with alkyldiammonium ions: a comparative studyFang, Guo-Sheng / Sun, Wen-Qi / Zhao, Wen-Xuan / Lin, Rui-Lian / Tao, Zhu / Liu, Jing-Xin et al. | 2015
- 680
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Design, synthesis and evaluation of N-aryl-glyoxamide derivatives as structurally novel bacterial quorum sensing inhibitorsNizalapur, Shashidhar / Kimyon, Önder / Biswas, Nripendra Nath / Gardner, Christopher R. / Griffith, Renate / Rice, Scott A. / Manefield, Mike / Willcox, Mark / Black, David StC. / Kumar, Naresh et al. | 2015
- 694
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Phosphinic acid-promoted addition reaction of isocyanides to (Z)-hydroximoyl chlorides: efficient synthesis of α-(hydroxyimino)amidesSoeta, Takahiro / Takashita, Suguru / Sakata, Yoko / Ukaji, Yutaka et al. | 2015
- 694
-
Phosphinic acid-promoted addition reaction of isocyanides to (Z)-hydroximoyl chlorides: efficient synthesis of a-(hydroxyimino)amidesSoeta, T. / Takashita, S. / Sakata, Y. / Ukaji, Y. et al. | 2016
- 701
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Molecular construction of HIV-gp120 discontinuous epitope mimics by assembly of cyclic peptides on an orthogonal alkyne functionalized TAC-scaffoldWerkhoven, P. R. / Elwakiel, M. / Meuleman, T. J. / Quarles van Ufford, H. C. / Kruijtzer, J. A. W. / Liskamp, R. M. J. et al. | 2015
- 711
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Oligomycins as inhibitors of K-Ras plasma membrane localisationSalim, A. A. / Tan, L. / Huang, X.-C. / Cho, K.-J. / Lacey, E. / Hancock, J. F. / Capon, R. J. et al. | 2015
- 716
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2-Aroylquinoline-5,8-diones as potent anticancer agents displaying tubulin and heat shock protein 90 (HSP90) inhibitionNepali, Kunal / Kumar, Sunil / Huang, Hsiang-Ling / Kuo, Fei-Chiao / Lee, Cheng-Hsin / Kuo, Ching-Chuan / Yeh, Teng-Kuang / Li, Yu-Hsuan / Chang, Jang-Yang / Liou, Jing-Ping et al. | 2015
- 724
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Isopropylmagnesium chloride-promoted unilateral addition of Grignard reagents to β-diketones: one-pot syntheses of β-tertiary hydroxyl ketones or 3-substituted cyclic-2-enonesYuan, Rui / Zhao, Dan / Zhang, Li-Yuan / Pan, Xiang / Yang, Yan / Wang, Pei / Li, Hong-Feng / Da, Chao-Shan et al. | 2015
- 724
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Isopropylmagnesium chloride-promoted unilateral addition of Grignard reagents to b-diketones: one-pot syntheses of b-tertiary hydroxyl ketones or 3-substituted cyclic-2-enonesYuan, R. / Zhao, D. / Zhang, L. Y. / Pan, X. / Yang, Y. / Wang, P. / Li, H. F. / Da, C. S. et al. | 2016
- 729
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A ligand-controlled switch of regioselectivity in ring-opening coupling of diarylmethylenecyclopropa[b]naphthalenes with Grignard reagentsCao, Jian / Huang, Xian / Wu, Luling et al. | 2015
- 738
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Selective recognition of neutral guests in an aqueous medium by a biomimetic calix[6]cryptamide receptorLascaux, Angélique / Leener, Gaël De / Fusaro, Luca / Topić, Filip / Rissanen, Kari / Luhmer, Michel / Jabin, Ivan et al. | 2015
- 738
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Selective recognition of neutral guests in an aqueous medium by a biomimetic calix[6]cryptamide receptorElectronic supplementary information (ESI) available: 1D and 2D NMR spectra of all new compounds, competitive NMR binding studies of 8 with Imi and Pyro and their behavior in acidic environment, refinement details of the structure solution and refinement of the crystal structures. CCDC 1428618 and 1428619. For ESI and crystallographic data in CIF or other electronic format see DOI: 10.1039/c5ob02067kLascaux, Angélique et al. | 2015
- 747
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Design and synthesis of simple, yet potent and selective non-ring-A pyripyropene A-based inhibitors of acyl-coenzyme A: cholesterol acyltransferase 2 (ACAT2)Zhan, Yang / Zhang, Xiao-Wei / Xiong, Ying / Li, Bo-Liang / Nan, Fa-Jun et al. | 2015
- 752
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Chiral bifunctional ferrocenylphosphine catalyzed highly enantioselective [3 + 2] cycloaddition reactionHu, Haiwen / Yu, Shuxian / Zhu, Linglong / Zhou, Lingxiu / Zhong, Weihui et al. | 2015
- 761
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Enantioselective organocatalytic oxidation of ketimineTakizawa, Shinobu / Kishi, Kenta / Abozeid, Mohamed Ahmed / Murai, Kenichi / Fujioka, Hiromichi / Sasai, Hiroaki et al. | 2015
- 768
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New electron-donor and -acceptor architectures from benzofurazans and sym-triaminobenzenes: intermediates, products and an unusual nitro group shiftMicheletti, G. / Boga, C. / Pafundi, M. / Pollicino, S. / Zanna, N. et al. | 2015
- 777
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A versatile approach to flavones via a one-pot Pd(ii)-catalyzed dehydrogenation/oxidative boron-Heck coupling sequence of chromanonesLee, Jun / Yu, Jihyun / Son, Seung Hwan / Heo, Jinyuk / Kim, Taelim / An, Ji-Young / Inn, Kyung-Soo / Kim, Nam-Jung et al. | 2015
- 785
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Correction: Multivalent presentation of carbohydrates by 314-helical peptide templates: synthesis, conformational analysis using CD spectroscopy and saccharide recognitionPawar, Nitin J. / Diederichsen, Ulf / Dhavale, Dilip. D. et al. | 2015
- 786
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Correction: One-pot synthesis of carbazoles via tandem C–C cross-coupling and reductive aminationGoo, Deuk-Young / Woo, Sang Kook et al. | 2015
- 787
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Back cover| 2015
- 4571
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Trifluoroacetic acid catalyzed highly regioselective bromocyclization of styrene-type carboxylic acidElectronic supplementary information (ESI) available. See DOI: 10.1039/c6ob00756bChen, Tao et al. | 2016
- 4576
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Design, synthesis, and in vitro evaluation of a fluorescently labeled irreversible inhibitor of the catalytic subunit of cAMP-dependent protein kinase (PKAC)Electronic supplementary information (ESI) available: Supplementary Fig. S1 and Tables S1 and S2, organic synthesis, characterization, and assay procedures. See DOI: 10.1039/c6ob00529bCoover, Robert A et al. | 2016
- 4582
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Rhodium-catalyzed asymmetric hydrogenation of unprotected -enamine phosphonatesElectronic supplementary information (ESI) available: Experimental procedures, NMR spectra of compounds. See DOI: 10.1039/c6ob00540cZhou, Ming et al. | 2016
- 4585
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Amino acid-promoted C-H alkylation with alkylboronic acids using a removable directing groupElectronic supplementary information (ESI) available. See DOI: 10.1039/c6ob00674dZhang, Yu et al. | 2016
- 4617
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Antimalarial activity of novel 4-cyano-3-methylisoquinoline inhibitors against Plasmodium falciparum: design, synthesis and biological evaluationElectronic supplementary information (ESI) available: Copies of the 1H and 13C NMR spectra of compounds 9-50. Counter screen of compounds 4, 12, 13, 23 and 25. Video S1. Live cell image sequence of a Plasmodium falciparum schizont-stage parasite treated with 10 M compound 25 showing egressing merozoites and their attempts to invade nearby erythrocytes. Some invasions were successful (white arrows) whilst some failed to penetrate (pink arrow) or could penetrate but not reseal their erythrocyte host (red arrow). Video S2. Live cell image sequence of a Plasmodium falciparum schizont-stage parasite treated with 10 M compound 25 showing egressing merozoites and their attempts to invade nearby erythrocytes. Some invasions were successful (white arrows) whilst some failed to penetrate (pink, yellow, orange and green arrows) or could penetrate but not reseal their erythrocyte host (red and blue arrows). See DOI: 10.1039/c5ob02517fBuskes, Melissa J et al. | 2016
- 4654
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PIDA-I2 mediated direct vicinal difunctionalization of olefins: iodoazidation, iodoetherification and iodoacyloxylationElectronic supplementary information (ESI) available: The file contains the 1H and 13C NMR spectra of the compounds. See DOI: 10.1039/c6ob00532bAchar, Tapas Kumar et al. | 2016
- 4664
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An efficient indenyl-derived phosphine ligand for the Suzuki-Miyaura coupling of sterically hindered aryl halidesElectronic supplementary information (ESI) available. See DOI: 10.1039/c6ob00096gLiu, Yan et al. | 2016
- 4669
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Efficient one-pot synthesis of amino-benzotriazolodiazocinone scaffolds via catalyst-free tandem Ugi-Huisgen reactionsElectronic supplementary information (ESI) available. See DOI: 10.1039/c6ob00438eBarlow, T. M. A et al. | 2016
- 4678
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ent-Abietane diterpenoids with anti-neuroinflammatory activity from the rare Chloranthaceae plant Chloranthus oldhamiiElectronic supplementary information (ESI) available: 1D/2D NMR and HRMS spectra of compounds 1-12 and 5a, the X-ray crystallographic data (CIF) of 1, and TDDFT ECD calculations for compounds 4 and 5. CCDC 1422696. For ESI and crystallographic data in CIF or other electronic format see DOI: 10.1039/c6ob00731gXiong, Juan et al. | 2016
- 4712
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Cation-halide transport through peptide pores containing aminopicolinic acidElectronic supplementary information (ESI) available: Detailed experimental procedures, characterization of compounds, analysis of fluorescence data, microscopy data, dynamic light scattering data. See DOI: 10.1039/c6ob00592fBasak, Debajyoti et al. | 2016
- 4718
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Exploring the divalent effect in fucosidase inhibition with stereoisomeric pyrrolidine dimersElectronic supplementary information (ESI) available: 1H and 13C-NMR spectra of new compounds, macromolecular X-ray data collection and refinement statistics for crystal structure determination and Lineweaver-Burk plots. See DOI: 10.1039/c6ob00647gHottin, Audrey et al. | 2016
- 4728
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Reversible and formaldehyde-mediated covalent binding of a bis-amino mitoxantrone analogue to DNAKonda, Shyam K et al. | 2016
- 4739
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Optimization and multigram scalability of a catalytic enantioselective borylative migration for the synthesis of functionalized chiral piperidinesElectronic supplementary information (ESI) available: 1H and 13C NMR spectra of new compounds and experimental procedures. See DOI: 10.1039/c6ob00685jKim, You-Ri et al. | 2016
- 4749
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Synthesis of imides via palladium-catalyzed decarboxylative amidation of -oxocarboxylic acids with secondary amidesElectronic supplementary information (ESI) available. See DOI: 10.1039/c6ob00676kXu, Ning et al. | 2016
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Rhodium-catalyzed C-C coupling reactions via double C-H activationLi, Shuai-Shuai et al. | 2016
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A fluorescent HTS assay for phosphohydrolases based on nucleoside 5-fluorophosphates: its application in screening for inhibitors of mRNA decapping scavenger and PDE-IElectronic supplementary information (ESI) available. See DOI: 10.1039/c6ob00492jBaranowski, M. R et al. | 2016
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Assessing histidine tags for recruiting deoxyribozymes to catalyze peptide and protein modification reactionsElectronic supplementary information (ESI) available. See DOI: 10.1039/c6ob00716cChu, Chih-Chi et al. | 2016