Discovery and pharmacological characterization of a selective delta opiate receptor antagonist (CP-646,777) (English)
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- New search for: Liras, Spiro
- New search for: McHardy, Stanton F.
- New search for: Allen, Martin P.
- New search for: Segelstein, Barb E.
- New search for: Heck, Steven D.
- New search for: Bryce, Dianne K.
- New search for: Schmidt, Anne W.
- New search for: O'Connor, Rebecca
- New search for: Vanase-Frawley, Michelle
- New search for: Callegari, Ernesto
- New search for: McLean, Stafford
- New search for: Liras, Spiro
- New search for: McHardy, Stanton F.
- New search for: Allen, Martin P.
- New search for: Segelstein, Barb E.
- New search for: Heck, Steven D.
- New search for: Bryce, Dianne K.
- New search for: Schmidt, Anne W.
- New search for: O'Connor, Rebecca
- New search for: Vanase-Frawley, Michelle
- New search for: Callegari, Ernesto
- New search for: McLean, Stafford
In:
MedChemComm
;
2
, 5
;
413-417
;
2011
- Article (Journal) / Electronic Resource
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Title:Discovery and pharmacological characterization of a selective delta opiate receptor antagonist (CP-646,777)
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Contributors:Liras, Spiro ( author ) / McHardy, Stanton F. ( author ) / Allen, Martin P. ( author ) / Segelstein, Barb E. ( author ) / Heck, Steven D. ( author ) / Bryce, Dianne K. ( author ) / Schmidt, Anne W. ( author ) / O'Connor, Rebecca ( author ) / Vanase-Frawley, Michelle ( author ) / Callegari, Ernesto ( author )
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Published in:MedChemComm ; 2, 5 ; 413-417
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Publisher:
- New search for: The Royal Society of Chemistry
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Publication date:2011-05-01
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Size:5 pages
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ISSN:
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Coden:
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DOI:
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Type of media:Article (Journal)
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Type of material:Electronic Resource
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Language:English
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Source:
Table of contents – Volume 2, Issue 5
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 339
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Front cover| 2011
- 340
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Inside front cover| 2011
- 341
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Contents| 2011
- 349
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Molecular obesity, potency and other addictions in drug discoveryHann, Michael M. et al. | 2011
- 356
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Computational ligand-based rational design: role of conformational sampling and force fields in model developmentShim, Jihyun / MacKerell, Jr., Alexander D. et al. | 2011
- 371
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Glycosylated porphyrin derivatives and their photodynamic activity in cancer cellsVedachalam, Seenuvasan / Choi, Bo-Hwa / Pasunooti, Kalyan Kumar / Ching, Kun Mei / Lee, Kijoon / Yoon, Ho Sup / Liu, Xue-Wei et al. | 2011
- 378
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Synthesis, in silico screening and bioevaluation of dispiro-cycloalkanones as antitubercular and mycobacterial NAD+-dependent DNA ligase inhibitorsTripathi, Rama P. / Pandey, Jyoti / Kukshal, Vandana / Ajay, Arya / Mishra, Mridul / Dube, Divya / Chopra, Deepti / Dwivedi, R. / Chaturvedi, Vinita / Ramachandran, Ravishankar et al. | 2011
- 385
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Synthesis and SAR studies of benzimidazole derivatives as melanin concentrating hormone receptor 1 (MCHR1) antagonists: Focus to detune hERG inhibitionSasmal, Pradip K. / Sasmal, Sanjita / Abbineni, Chandrasekhar / Venkatesham, B. / Rao, P. Tirumala / Roshaiah, M. / Khanna, Ish / Sebastian, V. J. / Suresh, J. / Singh, Manvendra P. et al. | 2011
- 390
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An approach to enzyme inhibition employing reversible boronate ester formationLeung, Ivanhoe K. H. / Brown Jr, Tom / Schofield, Christopher J. / Claridge, Timothy D. W. et al. | 2011
- 396
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Binding properties and biological characterization of new sugar-derived Ras ligandsSacco, Elena / Abraham, Sherwin J. / Palmioli, Alessandro / Damore, Gaetana / Bargna, Anna / Mazzoleni, Elisa / Gaponenko, Vadim / Vanoni, Marco / Peri, Francesco et al. | 2011
- 402
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trans-Stilbenoids: potent and selective inhibitors for human cytochrome P450 1B1Chun, Young-Jin / Lim, Chaemin / Ohk, Seul Ong / Lee, Ji Min / Lee, Jin Hee / Choi, Sun / Kim, Sanghee et al. | 2011
- 406
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Tacrine-mefenamic acid hybrids for inhibition of acetylcholinesteraseBornstein, Joshua J. / Eckroat, Todd J. / Houghton, Jacob L. / Jones, Christopher K. / Green, Keith D. / Garneau-Tsodikova, Sylvie et al. | 2011
- 413
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Discovery and pharmacological characterization of a selective delta opiate receptor antagonist (CP-646,777)Liras, Spiros / McHardy, Stanton F. / Allen, Martin P. / Segelstein, Barb E. / Heck, Steven D. / Bryce, Dianne K. / Schmidt, Anne W. / O'Connor, Rebecca / Vanase-Frawley, Michelle / Callegari, Ernesto et al. | 2011
- 418
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Inhibition of Pseudomonas aeruginosa biofilms with a glycopeptide dendrimer containing D-amino acidsJohansson, Emma M. V. / Kadam, Rameshwar U. / Rispoli, Gabriele / Crusz, Shanika A. / Bartels, Kai-Malte / Diggle, Stephen P. / Cámara, Miguel / Williams, Paul / Jaeger, Karl-Erich / Darbre, Tamis et al. | 2011
- 421
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Effective multi-strain inhibition of influenza virus by anionic gold nanoparticlesSametband, Matias / Shukla, Sourabh / Meningher, Tal / Hirsh, Shira / Mendelson, Ella / Sarid, Ronit / Gedanken, Aharon / Mandelboim, Michal et al. | 2011
- 424
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Structure–function study of gemini derivatives with two different side chains at C-20, Gemini-0072 and Gemini-0097Huet, Tiphaine / Maehr, Hubert / Lee, Hong Jin / Uskokovic, Milan R. / Suh, Nanjoo / Moras, Dino / Rochel, Natacha et al. | 2011
- 430
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Ester prodrugs of ciprofloxacin as DNA-gyrase inhibitors: synthesis, antiparasitic evaluation and docking studiesDubar, Faustine / Wintjens, René / Martins-Duarte, Érica S. / Vommaro, Rossiane C. / de Souza, Wanderley / Dive, Daniel / Pierrot, Christine / Pradines, Bruno / Wohlkonig, Alexandre / Khalife, Jamal et al. | 2011
- 436
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Edaravone containing isoindoline nitroxides for the potential treatment of cardiovascular ischaemiaWalker, James R. / Fairfull-Smith, Kathryn E. / Anzai, Kazunori / Lau, Shannen / White, Paul J. / Scammells, Peter J. / Bottle, Steven E. et al. | 2011
- 442
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MedChemWatch Issue 12 and Back cover| 2011