Design and synthesis of isothiocyanate‐containing hybrid androgen receptor (AR) antagonist to downregulate AR and induce ferroptosis in GSH–Deficient prostate cancer cells (English)
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In:
Chemical Biology & Drug Design
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97
, 5
;
1059-1078
;
2021
- Article (Journal) / Electronic Resource
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Title:Design and synthesis of isothiocyanate‐containing hybrid androgen receptor (AR) antagonist to downregulate AR and induce ferroptosis in GSH–Deficient prostate cancer cells
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Contributors:Qin, Zhihui ( author ) / Ou, Siyu ( author ) / Xu, Liping ( author ) / Sorensen, Kathleen ( author ) / Zhang, Yingxue ( author ) / Hu, Dan‐Ping ( author ) / Yang, Zhe ( author ) / Hu, Wen‐Yang ( author ) / Chen, Fei ( author ) / Prins, Gail S. ( author )
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Published in:Chemical Biology & Drug Design ; 97, 5 ; 1059-1078
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Publisher:
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Publication date:2021-05-01
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Size:20 pages
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ISSN:
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DOI:
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Type of media:Article (Journal)
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Type of material:Electronic Resource
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Language:English
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Keywords:
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Source:
Table of contents – Volume 97, Issue 5
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 1017
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A novel peptide isolated from garlic shows anticancer effect against leukemic cell lines via interaction with Bcl‐2 family proteinsRasaratnam, Karunaithas / Nantasenamat, Chanin / Phaonakrop, Narumon / Roytrakul, Sittiruk / Tanyong, Dalina et al. | 2021
- 1029
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Studying the helical conformations of aspereline peptidesBlanár, Eszter / Leitgeb, Balázs et al. | 2021
- 1038
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Ursolic and betulinic semisynthetic derivatives show activity against CQ‐resistant Plasmodium falciparum isolated from AmazoniaSol Sol de Medeiros, Daniel / Tasca Cargnin, Simone / Azevedo dos Santos, Ana Paula / de Souza Rodrigues, Moreno / Berton Zanchi, Fernando / Soares de Maria de Medeiros, Patrícia / de Almeida e Silva, Alexandre / Bioni Garcia Teles, Carolina / Baggio Gnoatto, Simone Cristina et al. | 2021
- 1048
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Discovery of drug‐like acetylcholinesterase inhibitors by rapid virtual screening of a 6.9 million compound databaseMiles, Jared A. / Ng, Jia Hui / Sreenivas, B. Yogi / Courageux, Charlotte / Igert, Alexandre / Dias, José / McGeary, Ross P. / Brazzolotto, Xavier / Ross, Benjamin P. et al. | 2021
- 1059
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Design and synthesis of isothiocyanate‐containing hybrid androgen receptor (AR) antagonist to downregulate AR and induce ferroptosis in GSH–Deficient prostate cancer cellsQin, Zhihui / Ou, Siyu / Xu, Liping / Sorensen, Kathleen / Zhang, Yingxue / Hu, Dan‐Ping / Yang, Zhe / Hu, Wen‐Yang / Chen, Fei / Prins, Gail S. et al. | 2021
- 1079
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Synergistic antifungal effects of curcumin derivatives as fungal biofilm inhibitors with fluconazoleDong, Huai‐Huai / Wang, Yuan‐Hua / Peng, Xue‐Mi / Zhou, He‐Yang / Zhao, Fei / Jiang, Yuan‐Ying / Zhang, Da‐Zhi / Jin, Yong‐Sheng et al. | 2021
- 1089
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W2476 represses TXNIP transcription via dephosphorylation of FOXO1 at Ser319Zhong, Li / Liu, Qing / Liu, Qiaofeng / Zhang, Shikai / Cao, Yongbing / Yang, Dehua / Wang, Ming‐Wei et al. | 2021
- 1100
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Secondary structure dependence of amyloid‐β(1–40) on simulation techniques and force field parametersCaliskan, Murat / Mandaci, Sunay Y. / Uversky, Vladimir N. / Coskuner‐Weber, Orkid et al. | 2021
- 1109
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Design, synthesis and biological evaluation of benz‐fused five‐membered heterocyclic compounds as tubulin polymerization inhibitors with anticancer activitiesKomuraiah, Buduma / Ren, Yichang / Xue, Mingming / Cheng, Binbin / Liu, Jin / Liu, Yao / Chen, Jianjun et al. | 2021
- 1117
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Design, synthesis, and biological evaluation of novel 4,4‐difluoro‐1‐methyl‐N, 6‐diphenyl‐5, 6‐dihydro‐4H‐pyrimido [4, 5‐b] [1, 2, 4] triazolo [4, 3‐d] [1, 4] diazepin‐8‐amine derivatives as potential BRD4 inhibitorsLi, Jiuhui / Zhang, Wenjie / Qiu, Qianqian / Zhou, Daoguang / Feng, Ziying / Tong, Zhenzhen / Wei, Jiaxin / Huang, Wenlong / Li, Jieming / Qian, Hai et al. | 2021
- i
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Cover ImageMiles, Jared A. / Ng, Jia Hui / Sreenivas, B. Yogi / Courageux, Charlotte / Igert, Alexandre / Dias, José / McGeary, Ross P. / Brazzolotto, Xavier / Ross, Benjamin P. et al. | 2021
- ii
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Issue Information| 2021