Structural Basis of Src Tyrosine Kinase Inhibition with a New Class of Potent and Selective Trisubstituted Purine‐based Compounds (English)
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In:
Chemical Biology & Drug Design
;
67
, 1
;
46-57
;
2006
- Article (Journal) / Electronic Resource
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Title:Structural Basis of Src Tyrosine Kinase Inhibition with a New Class of Potent and Selective Trisubstituted Purine‐based Compounds
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Contributors:Dalgarno, David ( author ) / Stehle, Thilo ( author ) / Narula, Surinder ( author ) / Schelling, Pierre ( author ) / Rose van Schravendijk, Marie ( author ) / Adams, Susan ( author ) / Andrade, Lawrence ( author ) / Keats, Jeff ( author ) / Ram, Mary ( author ) / Jin, Lei ( author )
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Published in:Chemical Biology & Drug Design ; 67, 1 ; 46-57
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Publisher:
- New search for: Blackwell Publishing Ltd
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Publication date:2006-01-01
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Size:12 pages
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ISSN:
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DOI:
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Type of media:Article (Journal)
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Type of material:Electronic Resource
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Language:English
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Source:
Table of contents – Volume 67, Issue 1
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 1
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Chemical Biology & Drug Design: Inaugural issue!Sawyer, Tomi K. et al. | 2006
- 2
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Overcoming Roadblocks in Lead Optimization: A Thermodynamic PerspectiveRuben, Adam J / Kiso, Yoshiaki / Freire, Ernesto et al. | 2006
- 5
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Structural Interaction Fingerprints: A New Approach to Organizing, Mining, Analyzing, and Designing Protein–Small Molecule ComplexesSingh, Juswinder / Deng, Zhan / Narale, Gaurav / Chuaqui, Claudio et al. | 2006
- 13
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Peptide, Peptidomimetic and Small‐molecule Drug Discovery Targeting HIV‐1 Host‐cell Attachment and Entry through gp120, gp41, CCR5 and CXCR4†Kazmierski, Wieslaw M. / Kenakin, Terry P. / Gudmundsson, Kristjan S. et al. | 2006
- 27
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Inhibition of Amyloid Fibril Formation by Polyphenols: Structural Similarity and Aromatic Interactions as a Common Inhibition MechanismPorat, Yair / Abramowitz, Adel / Gazit, Ehud et al. | 2006
- 38
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The Role of Water in Computational and Experimental Derivation of Binding Thermodynamics in SH2 DomainsGeroult, Sebastien / Virdee, Satpal / Waksman, Gabriel et al. | 2006
- 46
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Structural Basis of Src Tyrosine Kinase Inhibition with a New Class of Potent and Selective Trisubstituted Purine‐based CompoundsDalgarno, David / Stehle, Thilo / Narula, Surinder / Schelling, Pierre / Rose van Schravendijk, Marie / Adams, Susan / Andrade, Lawrence / Keats, Jeff / Ram, Mary / Jin, Lei et al. | 2006
- 58
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Structure‐based Optimization of MurF InhibitorsStamper, Geoffrey F. / Longenecker, Kenton L. / Fry, Elizabeth H. / Jakob, Clarissa G. / Florjancic, Alan S. / Gu, Yu‐Gui / Anderson, David D. / Cooper, Curt S. / Zhang, Tianyuan / Clark, Richard F. et al. | 2006
- 66
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Cellular Analysis of Disorazole C1 and Structure–Activity Relationship of Analogs of the Natural ProductWipf, Peter / Graham, Thomas H. / Vogt, Andreas / Sikorski, Rachel P. / Ducruet, Alexander P. / Lazo, John S. et al. | 2006
- 74
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The Discovery of Small Molecule Inhibitors of Neutral Endopeptidase. Structure–Activity Studies on Functionalized GlutaramidesMaw, Graham N. / Stobie, Alan / Planken, Simon / Pryde, David C. / Sanderson, Vivienne / Platts, Michelle Y. / Corless, Martin / Stacey, Peter / Wayman, Christopher / Van Der Graaf, Piet et al. | 2006
- 78
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Stability of Gold Nanoparticle‐Bound DNA toward Biological, Physical, and Chemical AgentsHan, Gang / Martin, Craig T. / Rotello, Vincent M. et al. | 2006
- 83
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Use of an Induced Fit Receptor Structure in Virtual ScreeningSherman, Woody / Beard, Hege S. / Farid, Ramy et al. | 2006
- 85
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A Chemogenomic Approach to Discovering Target‐Selective DrugsJanzen, William P. / Hodge, C. Nicholas et al. | 2006
- 87
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Biochemical Microarrays for Studying Chemical Biology Interaction: DiscoveryDotTM TechnologyHoriuchi, Kurumi Y. / Wang, Yuan / Ma, Haiching et al. | 2006
- 89
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Who's Who in Chemical Biology & Drug Design| 2006
- 96
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Calendar of Events| 2006