X-ray Crystal Structure and Binding Mode Analysis of Human S-Adenosylhomocysteine Hydrolase Complexed with Novel Mechanism-Based Inhibitors, Haloneplanocin A Analogues (Unknown)
- New search for: Lee, Kang Man
- New search for: Choi, Won Jun
- New search for: Lee, Yoonji
- New search for: Lee, Hyun Joo
- New search for: Zhao, Long Xuan
- New search for: Lee, Hyuk Woo
- New search for: Park, Jae Gyu
- New search for: Kim, Hea Ok
- New search for: Hwang, Kwang Yeon
- New search for: Heo, Yong-Seok
- New search for: Choi, Sun
- New search for: Jeong, Lak Shin
- New search for: Lee, Kang Man
- New search for: Choi, Won Jun
- New search for: Lee, Yoonji
- New search for: Lee, Hyun Joo
- New search for: Zhao, Long Xuan
- New search for: Lee, Hyuk Woo
- New search for: Park, Jae Gyu
- New search for: Kim, Hea Ok
- New search for: Hwang, Kwang Yeon
- New search for: Heo, Yong-Seok
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In:
Journal of Medicinal Chemistry
;
54
, 4
;
930-938
;
2011
- Article (Journal) / Electronic Resource
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Title:X-ray Crystal Structure and Binding Mode Analysis of Human S-Adenosylhomocysteine Hydrolase Complexed with Novel Mechanism-Based Inhibitors, Haloneplanocin A Analogues
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Additional title:J. Med. Chem.
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Contributors:Lee, Kang Man ( author ) / Choi, Won Jun ( author ) / Lee, Yoonji ( author ) / Lee, Hyun Joo ( author ) / Zhao, Long Xuan ( author ) / Lee, Hyuk Woo ( author ) / Park, Jae Gyu ( author ) / Kim, Hea Ok ( author ) / Hwang, Kwang Yeon ( author ) / Heo, Yong-Seok ( author )
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Published in:Journal of Medicinal Chemistry ; 54, 4 ; 930-938
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Publisher:
- New search for: American Chemical Society
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Publication date:2011-02-24
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ISSN:
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Coden:
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DOI:
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Type of media:Article (Journal)
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Type of material:Electronic Resource
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Language:Unknown
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Source:
Table of contents – Volume 54, Issue 4
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 915
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ATP-Binding Site of Bacterial Enzymes as a Target for Antibacterial Drug DesignŠkedelj, Veronika / Tomašić, Tihomir / Mašič, Lucija Peterlin / Zega, Anamarija et al. | 2011
- 930
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X-ray Crystal Structure and Binding Mode Analysis of Human S-Adenosylhomocysteine Hydrolase Complexed with Novel Mechanism-Based Inhibitors, Haloneplanocin A AnaloguesLee, Kang Man / Choi, Won Jun / Lee, Yoonji / Lee, Hyun Joo / Zhao, Long Xuan / Lee, Hyuk Woo / Park, Jae Gyu / Kim, Hea Ok / Hwang, Kwang Yeon / Heo, Yong-Seok et al. | 2011
- 939
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Development and Evaluation of Endothelin-A Receptor (Radio)Ligands for Positron Emission TomographyMichel, Kristin / Büther, Katrin / Law, Marilyn P. / Wagner, Stefan / Schober, Otmar / Hermann, Sven / Schäfers, Michael / Riemann, Burkhard / Höltke, Carsten / Kopka, Klaus et al. | 2011
- 949
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Synthesis and Evaluation of ^1^1C-Labeled Imidazo[2,1-b]benzothiazoles (IBTs) as PET Tracers for Imaging beta -Amyloid Plaques in Alzheimer's DiseaseYousefi, B.H. / Manook, A. / Drzezga, A. / Reutern, B.v. / Schwaiger, M. / Wester, H.-J. / Henriksen, G. et al. | 2011
- 949
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Synthesis and Evaluation of 11C-Labeled Imidazo[2,1-b]benzothiazoles (IBTs) as PET Tracers for Imaging β-Amyloid Plaques in Alzheimer’s DiseaseYousefi, Behrooz H. / Manook, André / Drzezga, Alexander / v. Reutern, Boris / Schwaiger, Markus / Wester, Hans-Jürgen / Henriksen, Gjermund et al. | 2011
- 957
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Probes for Narcotic Receptor Mediated Phenomena. 41. Unusual Inverse μ-Agonists and Potent μ-Opioid Antagonists by Modification of the N-Substituent in Enantiomeric 5-(3-Hydroxyphenyl)morphansCheng, Kejun / Lee, Yong Sok / Rothman, Richard B. / Dersch, Christina M. / Bittman, Ross W. / Jacobson, Arthur E. / Rice, Kenner C. et al. | 2011
- 970
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In Vivo Trypanosomicidal Activity of Imidazole- or Pyrazole-Based Benzo[g]phthalazine Derivatives against Acute and Chronic Phases of Chagas DiseaseSánchez-Moreno, Manuel / Sanz, Ana M. / Gómez-Contreras, Fernando / Navarro, Pilar / Marín, Clotilde / Ramírez-Macias, Inmaculada / Rosales, María Jose / Olmo, Francisco / Garcia-Aranda, Isabel / Campayo, Lucrecia et al. | 2011
- 980
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Synthesis and Pharmacological Activities of 6-Glycine Substituted 14-Phenylpropoxymorphinans, a Novel Class of Opioids with High Opioid Receptor Affinities and Antinociceptive PotenciesSpetea, Mariana / Windisch, Petra / Guo, Yan / Bileviciute-Ljungar, Indre / Schütz, Johannes / Asim, Muhammad Faheem / Berzetei-Gurske, Ilona P. / Riba, Pal / Kiraly, Kornel / Fürst, Susanna et al. | 2011
- 989
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Cationic Surfactants Derived from Lysine: Effects of Their Structure and Charge Type on Antimicrobial and Hemolytic ActivitiesColomer, A. / Pinazo, A. / Manresa, M. A. / Vinardell, M. P. / Mitjans, M. / Infante, M. R. / Pérez, L. et al. | 2011
- 1003
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Electron Paramagnetic Resonance (EPR) Study of Spin-Labeled Camptothecin Derivatives: A Different Look of the Ternary ComplexRicci, Antonio / Marinello, Jessica / Bortolus, Marco / Sánchez, Albert / Grandas, Anna / Pedroso, Enrique / Pommier, Yves / Capranico, Giovanni / Maniero, Anna Lisa / Zagotto, Giuseppe et al. | 2011
- 1010
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2-Aminothiazoles as Therapeutic Leads for Prion DiseasesGallardo-Godoy, Alejandra / Gever, Joel / Fife, Kimberly L. / Silber, B. Michael / Prusiner, Stanley B. / Renslo, Adam R. et al. | 2011
- 1022
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Analogues of σ Receptor Ligand 1-Cyclohexyl-4-[3-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]piperazine (PB28) with Added Polar Functionality and Reduced Lipophilicity for Potential Use as Positron Emission Tomography RadiotracersAbate, Carmen / Niso, Mauro / Lacivita, Enza / Mosier, Philip D. / Toscano, Annamaria / Perrone, Roberto et al. | 2011
- 1022
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Analogues of sigma Receptor Ligand 1-Cyclohexyl-4-[3-(5-methoxy-1,2,3,4-tetrahydronaphthaien-1-yl)propyl]-piperazine (PB28) with Added Polar Functionality and Reduced Lipophilicity for Potential Use as Positron Emission Tomography RadiotracersAbate, C. / Niso, M. / Lacivita, E. / Mosier, P.D. / Toscano, A. / Perrone, R. et al. | 2011
- 1033
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Evaluation of Quinazoline Analogues as Glucocerebrosidase Inhibitors with Chaperone ActivityMarugan, Juan J. / Zheng, Wei / Motabar, Omid / Southall, Noel / Goldin, Ehud / Westbroek, Wendy / Stubblefield, Barbara K. / Sidransky, Ellen / Aungst, Ronald A. / Lea, Wendy A. et al. | 2011
- 1059
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Acyloxy Nitroso Compounds as Nitroxyl (HNO) Donors: Kinetics, Reactions with Thiols, and Vasodilation PropertiesShoman, Mai E. / DuMond, Jenna F. / Isbell, T. S. / Crawford, J. H. / Brandon, Angela / Honovar, Jaideep / Vitturi, Dario A. / White, C. R. / Patel, R. P. / King, S. Bruce et al. | 2011
- 1071
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Discovery and Biological Characterization of (2R,4S)-1′-Acetyl-N-{(1R)-1-[3,5-bis(trifluoromethyl)phenyl]ethyl}-2-(4-fluoro-2-methylphenyl)-N-methyl-4,4′-bipiperidine-1-carboxamide as a New Potent and Selective Neurokinin 1 (NK1) Receptor Antagonist Clinical CandidateDi Fabio, Romano / Alvaro, Giuseppe / Griffante, Cristiana / Pizzi, Domenica A. / Donati, Daniele / Mattioli, Mario / Cimarosti, Zadeo / Guercio, Giuseppe / Marchioro, Carla / Provera, Stefano et al. | 2011
- 1080
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Biotin Ergopeptide Probes for Dopamine ReceptorsVendrell, Marc / Molero, Anabel / González, Sergio / Pérez-Capote, Kamil / Lluis, Carme / McCormick, Peter J. / Franco, Rafael / Cortés, Antoni / Casadó, Vicent / Albericio, Fernando et al. | 2011
- 1091
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Convergent Evolution-Guided Design of Antimicrobial Peptides Derived from Influenza A Virus HemagglutininZhu, Shunyi / Aumelas, André / Gao, Bin et al. | 2011
- 1096
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Development of Non-Peptide Ligands of Growth Factor Receptor-Bound Protein 2-Src Homology 2 Domain Using Molecular Modeling and NMR SpectroscopyOrcajo-Rincón, Ángel L. / Ortega-Gutiérrez, Silvia / Serrano, Pedro / Torrecillas, Ivan R. / Wüthrich, Kurt / Campillo, Mercedes / Pardo, Leonardo / Viso, Alma / Benhamú, Bellinda / López-Rodríguez, María L. et al. | 2011
- 1101
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3-Thiomorpholin-8-oxo-8H-acenaphtho[1,2-b]pyrrole-9-carbonitrile (S1) Based Molecules as Potent, Dual Inhibitors of B-Cell Lymphoma 2 (Bcl-2) and Myeloid Cell Leukemia Sequence 1 (Mcl-1): Structure-Based Design and Structure−Activity Relationship StudiesZhang, Zhichao / Wu, Guiye / Xie, Feibo / Song, Ting / Chang, Xilong et al. | 2011
- 1106
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Discovery, Synthesis, and Structure−Activity Relationship Development of a Series of N-(4-Acetamido)phenylpicolinamides as Positive Allosteric Modulators of Metabotropic Glutamate Receptor 4 (mGlu4) with CNS Exposure in RatsEngers, Darren W. / Field, Julie R. / Le, Uyen / Zhou, Ya / Bolinger, Julie D. / Zamorano, Rocio / Blobaum, Anna L. / Jones, Carrie K. / Jadhav, Satyawan / Weaver, C. David et al. | 2011